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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50169467
(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
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Affinity Data
Ki: 2.30nM
Assay Description:
Inhibitory constant against human sst5 receptor at a dose of 10 uM
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W66MH6
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50169467
(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
copy SMILES
copy InChI
Affinity Data
Ki: 5.60nM
Assay Description:
Inhibitory constant against human sst2 receptor at a dose of 10 uM
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W66MH6
PubMed
Target
Somatostatin receptor type 5
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50169467
(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
copy SMILES
copy InChI
Affinity Data
EC50: 52nM
Assay Description:
Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptor
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W66MH6
PubMed
Target
Somatostatin receptor type 2
(Homo sapiens (Human))
Institut Henri Beaufour
Curated by
ChEMBL
Ligand
BDBM50169467
(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
copy SMILES
copy InChI
Affinity Data
EC50: 6.30nM
Assay Description:
Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptor
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2W66MH6
PubMed