Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetSomatostatin receptor type 5(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)copy SMILEScopy InChI
Affinity DataKi:  2.30nMAssay Description:Inhibitory constant against human sst5 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66MH6PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)copy SMILEScopy InChI
Affinity DataKi:  5.60nMAssay Description:Inhibitory constant against human sst2 receptor at a dose of 10 uMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66MH6PubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)copy SMILEScopy InChI
Affinity DataEC50:  52nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66MH6PubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institut Henri Beaufour

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)copy SMILEScopy InChI
Affinity DataEC50:  6.30nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66MH6PubMed