Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetMelanocortin receptor 3(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217773(CHEMBL428903 | N-(2-amino-ethyl)-4-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  2.70E+3nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC3 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocyte-stimulating hormone receptor(Mus musculus)
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217773(CHEMBL428903 | N-(2-amino-ethyl)-4-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of [125I]NDP-MSH from MC1 receptor in mouse B16 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217773(CHEMBL428903 | N-(2-amino-ethyl)-4-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC4 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed
TargetMelanocortin receptor 5(Homo sapiens (Human))
Uppsala University

Curated by ChEMBL
LigandPNGBDBM50217773(CHEMBL428903 | N-(2-amino-ethyl)-4-(1H-indol-3-yl)...)copy SMILEScopy InChI
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of [125I]NDP-MSH from human recombinant MC5 receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X066Q5PubMed