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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
G protein-coupled receptor kinase 5
(Homo sapiens (Human))
Korea Research Institute of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50444125
(CHEMBL3093150)
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copy InChI
Affinity Data
IC50: 810nM
Assay Description:
Inhibition of GRK-5 (unknown origin) preincubated with enzyme for 10 mins before adding peptide substrate and ATP measured after 1 hr by LANCE-TR-FRE...
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2SX6FPP
PubMed
Target
Beta-adrenergic receptor kinase 1
(Homo sapiens (Human))
Korea Research Institute of Chemical Technology
Curated by
ChEMBL
Ligand
BDBM50444125
(CHEMBL3093150)
copy SMILES
copy InChI
Affinity Data
IC50: 5.30E+3nM
Assay Description:
Inhibition of GRK-2 (unknown origin) preincubated with enzyme for 10 mins before adding peptide substrate and ATP measured after 1 hr by LANCE-TR-FRE...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2SX6FPP
PubMed