Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)copy SMILEScopy InChI
Affinity DataKi:  424nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q24Q7SGJPubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Binding affinity towards Thromboxane A2/ Prostaglandin H2 receptor in human platelet membranes using [125I]- as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B56KB7PubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Medical University of South Carolina

Curated by PDSP Ki Database
LigandPNGBDBM81947(CAS_113243-00-8 | L-657926)copy SMILEScopy InChI
Affinity DataIC50: 11.2nMAssay Description:Binding affinity towards Thromboxane A2/ Prostaglandin H2 receptor in human platelet membranes using [125I]- as the radioligand.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2B56KB7PubMed