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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Thromboxane-A synthase
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50283052
((Z)-7-[(2R,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
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Affinity Data
IC50: 32nM
Assay Description:
In vitro inhibition of the compound against thromboxane synthase
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2C53KS7
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
TBA
Curated by
ChEMBL
Ligand
BDBM50283052
((Z)-7-[(2R,3R,4R)-4-(Biphenyl-4-ylmethoxy)-2-pyrid...)
copy SMILES
copy InChI
Affinity Data
IC50: 795nM
Assay Description:
In vitro thromboxane receptor antagonist against U-46619 induced aggregation of washed human platelets
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2C53KS7