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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Thromboxane-A synthase
(Homo sapiens (Human))
University of Innsbruck
Curated by
ChEMBL
Ligand
BDBM50053753
(5-[1-Phenyl-1-pyridazin-3-yl-meth-(E)-ylideneamino...)
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Affinity Data
IC50: 1.00E+5nM
Assay Description:
TXA2 synthetase inhibition measured by the inhibition of TXB2 formation by human gel-filtered platelets incubated with [14C]-arachidonic acid
More data for this Ligand-Target Pair
Target Info
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2ZP456G
PubMed
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
University of Innsbruck
Curated by
ChEMBL
Ligand
BDBM50053753
(5-[1-Phenyl-1-pyridazin-3-yl-meth-(E)-ylideneamino...)
copy SMILES
copy InChI
Affinity Data
IC50: 1.04E+5nM
Assay Description:
TXA2 receptor antagonism, measured by the displacement of [3H]SQ29,548 from the PGH-2/TXA-2 receptor on human platelets
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
BindingDB Entry DOI:
10.7270/Q2ZP456G
PubMed