Home
About
Info
Download
WebServices
Contact
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
Thromboxane A2 receptor
(Homo sapiens (Human))
Pharmacia-Farmitalia Carlo Erba
Curated by
ChEMBL
Ligand
BDBM50037732
(5-[1-Cyclohexyl-2-imidazol-1-yl-3-(4-trifluorometh...)
copy SMILES
copy InChI
Affinity Data
IC50: 50nM
Assay Description:
In vitro thromboxane-A2 receptor binding affinity to displace by 50% [3H]-SQ 29548 binding from washed human platelets
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2C24VFD
PubMed
Target
Thromboxane-A synthase
(Rattus norvegicus)
Pharmacia-Farmitalia Carlo Erba
Curated by
ChEMBL
Ligand
BDBM50037732
(5-[1-Cyclohexyl-2-imidazol-1-yl-3-(4-trifluorometh...)
copy SMILES
copy InChI
Affinity Data
IC50: 900nM
Assay Description:
In vitro inhibition of thromboxane-A2 synthase in rat whole blood during clotting at 37 degrees centigrade
More data for this Ligand-Target Pair
Target Info
Reactome pathway
KEGG
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
BindingDB Entry DOI:
10.7270/Q2C24VFD
PubMed