Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetCholecystokinin(RAT)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)copy SMILEScopy InChI
Affinity DataKi:  1.40nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K05PubMed
TargetGABA(A) receptor-associated protein(GUINEA PIG)
Merck Sharp & Dohme Research Laboratories

Curated by PDSP Ki Database
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445K05PubMed
TargetCholecystokinin receptor type A(RAT)
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to cholecystokinin A receptor from rat pancreatic tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1S9KPubMed
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)copy SMILEScopy InChI
Affinity DataIC50: 650nMAssay Description:Half-maximal inhibition of [125I]gastrin binding to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1S9KPubMed
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Merck Sharp& Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50019219(CCK antagonist synthetic 20 | CHEMBL70456 | {3-[(1...)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-8(+) binding to cholecystokinin receptor from guinea pig brain tissueMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PG1S9KPubMed