Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
National Cancer Institute-CRO

Curated by ChEMBL
LigandPNGBDBM50144747(CHEMBL3763517)copy SMILEScopy InChI
Affinity DataKi:  5.46E+3nMAssay Description:Competitive inhibition of human LDH5 meaured for 3 mins in presence of pyruvate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27X41PubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
National Cancer Institute-CRO

Curated by ChEMBL
LigandPNGBDBM50144747(CHEMBL3763517)copy SMILEScopy InChI
Affinity DataKi:  1.51E+4nMAssay Description:Competitive inhibition of human LDH1 meaured for 3 mins in presence of pyruvate by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27X41PubMed
TargetL-lactate dehydrogenase B chain(Homo sapiens (Human))
National Cancer Institute-CRO

Curated by ChEMBL
LigandPNGBDBM50144747(CHEMBL3763517)copy SMILEScopy InChI
Affinity DataKi:  2.32E+4nMAssay Description:Competitive inhibition of human LDH1 meaured for 3 mins in presence of NADH by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27X41PubMed
TargetL-lactate dehydrogenase A chain(Homo sapiens (Human))
National Cancer Institute-CRO

Curated by ChEMBL
LigandPNGBDBM50144747(CHEMBL3763517)copy SMILEScopy InChI
Affinity DataKi:  5.60E+4nMAssay Description:Competitive inhibition of human LDH5 meaured for 3 mins in presence of NADH by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B27X41PubMed