Found 30 Enz. Inhib. hit(s) with Target = 'Beta-adrenergic receptor kinase 2' 
Affinity DataIC50: 0.00900nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0190nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0240nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0480nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0650nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.144nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.380nMAssay Description:ADRB2 IC50 from binding assay(nM), Determined using the Tag-lite Adrenoceptor Beta2 receptor ligand binding assay.More data for this Ligand-Target Pair
Affinity DataIC50: 0.650nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.80nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 4.30nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 5.40nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human full length GST-tagged GRK3 expressed in baculovirus using ulight topo2alpha as substrate preincubated for 60 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Inhibition of GRK3-mediated bovine tubulin phosphorylation by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 850nMAssay Description:Inhibition of human GRK3 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 861nMAssay Description:Inhibition of human GRK3 using casein as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 6.10E+3nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK3 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK3 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK3 using casein as substrate in presence of [gamma33P]ATP by radiometric hotspot kinase assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full length human GRK3 using casein as substrate after 40 mins in presence of [gamma-33ATP] by radiometric scintillation co...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human GRK3 using casein as substrateMore data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 1.16E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 2.26E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 3.04E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
TargetBeta-adrenergic receptor kinase 2(Bos taurus)
Universit£ degli Studi di Messina
Curated by ChEMBL
Universit£ degli Studi di Messina
Curated by ChEMBL
Affinity DataIC50: 5.55E+4nMAssay Description:Inhibition of recombinant bovine GRK3 expressed in Sf9 insect cells assessed as decrease in phosphorylation of urea-washed bovine rod outer segments ...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant full length human GST-tagged GRK3 expressed in baculovirus expression system using serine/threonine-16 peptide as substrate...More data for this Ligand-Target Pair
