Compile Data Set for Download or QSAR
Found 11 Enz. Inhib. hit(s) with Target = 'Bromodomain testis-specific protein [287-359]'
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM205429( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...)copy SMILEScopy InChI
Affinity DataIC50: 217nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM50103503(CHEMBL2393130 | US11117865, Compound RVX-208)copy SMILEScopy InChI
Affinity DataIC50: 708nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM518731(US11117865, Compound ZL0590)copy SMILES
Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM518731(US11117865, Compound ZL0590)copy SMILES
Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM518799(US11117865, Compound ZL0591)copy SMILES
Affinity DataIC50: 1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM518799(US11117865, Compound ZL0591)copy SMILES
Affinity DataIC50: 1.95E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM50370182(CHEMBL4176038 | US11117865, Compound ZL0420)copy SMILEScopy InChI
Affinity DataIC50: 2.78E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM50370181(CHEMBL4159382 | US11117865, Compound ZL0454)copy SMILEScopy InChI
Affinity DataIC50: 3.08E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM50527819(CHEMBL4557050 | US11117865, Compound ZL0516)copy SMILEScopy InChI
Affinity DataIC50: 3.18E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent
TargetBromodomain testis-specific protein [287-359](Homo sapiens (Human))TBA
LigandPNGBDBM518854(US11117865, Compound ZL0497)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TT4V40US Patent