Compile Data Set for Download or QSAR
Found 483 Enz. Inhib. hit(s) with Target = 'Cyclin-G-associated kinase'
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50546116(CHEMBL4797973)copy SMILES
Affinity DataKi:  1.5nMAssay Description:Binding affinity to GAK (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21J9FC5PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50524284(CHEMBL4443342)copy SMILEScopy InChI
Affinity DataKi:  3.10nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50537138(CHEMBL4531690)copy SMILEScopy InChI
Affinity DataKi:  3.80nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50537139(CHEMBL4535001)copy SMILEScopy InChI
Affinity DataKi:  49nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50184765(CHEMBL3823499)copy SMILEScopy InChI
Affinity DataKi:  220nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511378(CHEMBL4470026)copy SMILEScopy InChI
Affinity DataKi:  360nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511379(CHEMBL4447403)copy SMILEScopy InChI
Affinity DataKi:  510nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511398(CHEMBL4582326)copy SMILEScopy InChI
Affinity DataKi:  580nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511384(CHEMBL4561238)copy SMILEScopy InChI
Affinity DataKi:  780nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511385(CHEMBL4534959)copy SMILEScopy InChI
Affinity DataKi:  870nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511394(CHEMBL4552310)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511373(CHEMBL4571548)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511376(CHEMBL4516665)copy SMILEScopy InChI
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511397(CHEMBL4452939)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511383(CHEMBL4531680)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50273541(CHEMBL516312 | N-(5-(4-cyanophenyl)-1H-pyrrolo[2,3...)copy SMILEScopy InChI
Affinity DataKi:  1.75E+3nMAssay Description:Binding affinity to biotinylated GAK (unknown origin) incubated for 1.5 hrs by fluorescent tracer dependent TR-FRET based binding displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5XMRPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50524287(CHEMBL4462395)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511380(CHEMBL4452360)copy SMILEScopy InChI
Affinity DataKi:  2.60E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511400(CHEMBL4535040)copy SMILEScopy InChI
Affinity DataKi:  2.90E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511396(CHEMBL4472438)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511399(CHEMBL4542463)copy SMILEScopy InChI
Affinity DataKi:  3.20E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511374(CHEMBL4522276)copy SMILEScopy InChI
Affinity DataKi:  3.90E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511395(CHEMBL4473140)copy SMILEScopy InChI
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511375(CHEMBL4593649)copy SMILEScopy InChI
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50511377(CHEMBL4534571)copy SMILEScopy InChI
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of Alexafluor labelled kinase tracer236 from biotinylated C-terminal Avi-tagged GAK kinase domain (12 to 347 residues) (unknown origin) ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC8669PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50516677(CHEMBL4514780)copy SMILEScopy InChI
Affinity DataKi:  8.20E+3nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50524288(CHEMBL4518437)copy SMILEScopy InChI
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity to C-terminal AVI-tagged GAK (unknown origin) (12 to 347 residues) expressed in Escherichia coli after 1.5 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50537138(CHEMBL4531690)copy SMILEScopy InChI
Affinity DataIC50: 0.0600nMAssay Description:Displacement of fluorescent tracer from N-terminus of human GAK expressed in HEK293T cells after 2 hrs by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50332294(CHEMBL1287853 | N-tert-butyl-3-(5-methyl-2-(4-(2-(...)copy SMILEScopy InChI
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q801KPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562897(CHEMBL4740761)copy SMILES
Affinity DataIC50: 2.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM6503(4-Anilino-3-cyanoquinoline deriv. 4 | 6,7-dimethox...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMAssay Description:Inhibition of tracer 5 binding to human N-terminal nano luciferase-fused GAK expressed in HEK293 cells measured after 2 hrs by nanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4NVJPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562898(CHEMBL4778276)copy SMILES
Affinity DataIC50: 3.20nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562894(CHEMBL4762694)copy SMILES
Affinity DataIC50: 3.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562893(CHEMBL4764705)copy SMILES
Affinity DataIC50: 7.70nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562895(CHEMBL4794323)copy SMILES
Affinity DataIC50: 8.80nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50516677(CHEMBL4514780)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Displacement of fluorescent tracer from N-terminus of human GAK expressed in HEK293T cells after 2 hrs by NanoBRET target engagement assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28919C7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50362781(1256580-46-7 | AF802 | Alecensa | Alectinib | CH54...)copy SMILEScopy InChI
Affinity DataIC50: 10nMAssay Description:Inhibition of human GAKMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KK9GG7PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 11nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562914(CHEMBL4745919)copy SMILES
Affinity DataIC50: 12nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562913(CHEMBL4745028)copy SMILES
Affinity DataIC50: 13nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562905(CHEMBL4800032)copy SMILES
Affinity DataIC50: 14nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562896(CHEMBL4779229)copy SMILES
Affinity DataIC50: 17nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50538885(CHEMBL4646895)copy SMILEScopy InChI
Affinity DataIC50: 22nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM6511(4-Anilinoquinoline deriv. 8 | 6,7-dimethoxy-N-(3,4...)copy SMILEScopy InChI
Affinity DataIC50: 23nMAssay Description:Inhibition of tracer 5 binding to human N-terminal nano luciferase-fused GAK expressed in HEK293 cells measured after 2 hrs by nanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4NVJPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50538901(CHEMBL4642467)copy SMILEScopy InChI
Affinity DataIC50: 24nMAssay Description:Inhibition of tracer 222 binding to recombinant human GST-tagged GAK (1 to 329 residues) expressed in insect cells incubated for 1 hr by Lanthascreen...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TM7FNTPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50538901(CHEMBL4642467)copy SMILEScopy InChI
Affinity DataIC50: 24nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q801KPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50524281(CHEMBL4440586)copy SMILEScopy InChI
Affinity DataIC50: 31nMAssay Description:Inhibition of tracer 5 binding to human N-terminal nano luciferase-fused GAK expressed in HEK293 cells measured after 2 hrs by nanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RJ4NVJPubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562907(CHEMBL4752286)copy SMILES
Affinity DataIC50: 35nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM50562908(CHEMBL4784439)copy SMILES
Affinity DataIC50: 37nMAssay Description:Inhibition of tracer 222 binding to GAK (unknown origin) incubated for 1 hr by Lanthascreen TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R78JZ2PubMed
TargetCyclin-G-associated kinase(Homo sapiens (Human))TBA
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)copy SMILEScopy InChI
Affinity DataIC50: 38nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q801KPubMed
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