Affinity DataIC50: 5.60nMAssay Description:Inhibition of human DAPK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.30nMAssay Description:Inhibition of human DAPK2 using KKLNRTLSFAEPG as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of Dapk2 (unknown origin) by quantitative PCRMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 570nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 830nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
Affinity DataIC50: 6.34E+3nMAssay Description:Compound was tested for the inhibitory constant for adenosine deaminase (ADA)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of DAPK2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant full length human DAPK2 using Calmodulin as substrate incubated 40 mins in presence of [gamma-33ATP] by radiometric scintil...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human DAPK2 using [KKLNRTLSFAEPG] as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
Affinity DataIC50: 5.50E+4nMAssay Description:Inhibition of human DAPK2More data for this Ligand-Target Pair
In DepthDetails
Affinity DataKd: 2.70E+3nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Kinase inhibitors are a new class of therapeutics with a propensity to inhibit multiple targets. The biological consequences of multi-kinase activity...More data for this Ligand-Target Pair
Affinity DataKd: 610nMAssay Description:Average Binding Constant for DAPK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Average Binding Constant for DAPK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 3.20E+3nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 63nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 1.60nMAssay Description:Binding constant for full-length DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 890nMAssay Description:Binding constant for full-length DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 470nMAssay Description:Average Binding Constant for DAPK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: 2.60E+3nMAssay Description:Average Binding Constant for DAPK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to DAPK2More data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 930nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 62nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 29nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: >1.00E+4nMAssay Description:Binding constant for DAPK2 kinase domainMore data for this Ligand-Target Pair