Compile Data Set for Download or QSAR
Found 71 Enz. Inhib. hit(s) with Target = 'Disintegrin and metalloproteinase domain-containing protein 9'
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50265157((6S,7S)-N-hydroxy-5-methyl-6-(4-(5-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of recombinant human C-terminal His10-tagged ADAM9 (Ala206 to Asp697 residues) expressed in mouse cells using McaPLAQAV-Dpa-RSSSR-NH2 as s...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M688JPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50313818(5-((5-methoxy-3-oxo-1H-indazol-2(3H)-yl)methyl)-5-...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of ADAM9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2F76CQ9PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:In vitro inhibition of A disintegrin and metalloproteinase domain 9 (ADAM9)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM912((3S,4S)-3-hydroxy-4-[(2S)-2-[(3S,4S)-3-hydroxy-6-m...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2PXPPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Inhibition of ADAM9 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2PXPPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109614(CHEMBL353536 | [4-(2-Ethoxy-ethoxy)-phenyl]-(3-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109630((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50181008((S)-N-hydroxy-4-(4-(4-hydroxybut-2-ynyloxy)phenyls...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29W0DC8US Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50181008((S)-N-hydroxy-4-(4-(4-hydroxybut-2-ynyloxy)phenyls...)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAM9 and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TM78ZSUS Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM175095(US9115102, Apratastat)copy SMILEScopy InChI
Affinity DataIC50: 85nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5CRVUS Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50453825(CHEMBL4215407 | US10556883, Compound 19a)copy SMILEScopy InChI
Affinity DataIC50: 90nMAssay Description:Inhibition of ADAM9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9FPHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109631((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109610((7-Amino-3-hydroxycarbamoyl-3,4-dihydro-1H-isoquin...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50370191(CHEMBL366478)copy SMILEScopy InChI
Affinity DataIC50: 230nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109635((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109629((4-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109628((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 370nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109637(4-[Ethoxy-(4-methoxy-phenyl)-phosphinoyl]-3-hydrox...)copy SMILEScopy InChI
Affinity DataIC50: 430nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50453823(CHEMBL4208519 | US10556883, Compound 19d)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:Inhibition of ADAM9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9FPHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109634((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109624((6-Hydroxycarbamoyl-6,7-dihydro-4H-thieno[3,2-c]py...)copy SMILEScopy InChI
Affinity DataIC50: 520nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109616((7-Hydroxycarbamoyl-7,8-dihydro-5H-pyrido[3,4-b]py...)copy SMILEScopy InChI
Affinity DataIC50: 560nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109625((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 660nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109623((4-Amino-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-1...)copy SMILEScopy InChI
Affinity DataIC50: 660nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109613((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 700nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109633((3-Hydroxycarbamoyl-1,3,4,9-tetrahydro-beta-carbol...)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109627((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 810nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109632((3-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 830nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109640((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 890nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109611((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 910nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109612((2-Fluoro-phenyl)-(3-hydroxycarbamoyl-3,4-dihydro-...)copy SMILEScopy InChI
Affinity DataIC50: 1.06E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109615((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109622((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109639((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109621(CHEMBL425316 | [4-(4-Amino-phenoxy)-phenyl]-(3-hyd...)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109636((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109626(Biphenyl-4-yl-(3-hydroxycarbamoyl-3,4-dihydro-1H-i...)copy SMILEScopy InChI
Affinity DataIC50: 1.96E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109620((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 2.24E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109638((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM379557(US9926281, Compound 36)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of ADAM-9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM113589(US8633196, 19 | US9365529, 19)copy SMILEScopy InChI
Affinity DataIC50: 3.05E+3nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29W0DC8US Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109618((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 3.11E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM175076(US9115102, Ex2)copy SMILEScopy InChI
Affinity DataIC50: 3.25E+3nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5CRVUS Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50109617((3-Hydroxycarbamoyl-3,4-dihydro-1H-isoquinolin-2-y...)copy SMILEScopy InChI
Affinity DataIC50: 3.56E+3nMAssay Description:Inhibition of the heparin binding epidermal growth factor (HB-EGF) release from fibrosarcoma HT1080 transfectants expressing alkaline phosphate (AP) ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2XK8G9QPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50203527((6S,7S)-methyl 7-(hydroxycarbamoyl)-6-(4-phenyl-1,...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ADAM9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD4WM2PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50265157((6S,7S)-N-hydroxy-5-methyl-6-(4-(5-(trifluoromethy...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of ADAM9More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JD4WM2PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50575718(CHEMBL4873384)copy SMILES
Affinity DataIC50: 8.45E+3nMAssay Description:Inhibition of ADAM-9 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VBMPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM113588(US8633196, 18 | US9365529, 18)copy SMILEScopy InChI
Affinity DataIC50: 9.25E+3nMAssay Description:The molecules are dose-response tested on the following enzymes: MMP1, MMP3, MMP9, ADAM9 and ADAM10, according to the same protocol as that described...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29W0DC8US Patent
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM50236675(CHEMBL4102106)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of ADAM9 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28S4S59PubMed
TargetDisintegrin and metalloproteinase domain-containing protein 9(Homo sapiens (Human))
University of Notre Dame

Curated by ChEMBL
LigandPNGBDBM175083(US9115102, Ex14 | US9115102, Ex24)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:The molecules are tested in dose-response studies on the following enzymes MMP1, MMP3, MMP9, ADAMS and ADAM10 according to the same protocol as that ...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q21V5CRVUS Patent
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