Compile Data Set for Download or QSAR
Found 440 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1'
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  5nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232884(CHEMBL4060962)copy SMILEScopy InChI
Affinity DataKi:  18nMAssay Description:Displacement of [3H]strychnine from glycine receptor alpha 1 in rat brain synaptic membranesMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  23nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232885(CHEMBL4089150)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232888(CHEMBL4096857)copy SMILEScopy InChI
Affinity DataKi:  67nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50570357(CHEMBL4865147)copy SMILES
Affinity DataKi:  81nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PV6PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50510757(CHEMBL4518537)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataKi:  123nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataKi:  189nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50570358(CHEMBL4855686)copy SMILES
Affinity DataKi:  204nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PV6PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232897(CHEMBL4068867)copy SMILEScopy InChI
Affinity DataKi:  241nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataKi:  370nMAssay Description:Displacement of [3H]strychnine from recombinant human glycine receptor alpha 1 expressed in HEK293 cell membranes after 30 mins by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50570355(CHEMBL4873527)copy SMILES
Affinity DataKi:  436nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PV6PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50510756(CHEMBL4447664)copy SMILEScopy InChI
Affinity DataKi:  741nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2571GB7PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50570356(CHEMBL4864603)copy SMILES
Affinity DataKi:  977nMAssay Description:Displacement of [3H]strychnine from human glycine receptor subunit alpha-1 expressed in HEK293 cell membranes preincubated for 30 mins followed by [3...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PV6PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50022784((R)-N-methyl-3-phenyl-3-(o-tolyloxy)propan-1-amine...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6W98PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M648WPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M648WPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM84745(CAS_136434-34-9 | DULOXETINE | LY-248686 | LY24868...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M648WPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM82071(CAS_93413-69-5 | CAS_99300-78-4 | NSC_62923 | VENL...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25M648WPubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50022784((R)-N-methyl-3-phenyl-3-(o-tolyloxy)propan-1-amine...)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GQ6W98PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50133817(4-(3-Chloro-pyridin-2-yl)-piperazine-1-carboxylic ...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3CX5PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM22913(CHEMBL1237146 | CHEMBL498770 | Iodophenpropit | {[...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5F64PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM22869(6-chloro-10-(4-methylpiperazin-1-yl)-2,9-diazatric...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ865XPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ865XPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM81790(Amisulpride | CAS_71675-85-9 | NSC_2159 | US101672...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2NZ865XPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM22914(CHEMBL260374 | N-cyclohexyl-4-(1H-imidazol-5-yl)pi...)copy SMILEScopy InChI
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZK5F64PubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)copy SMILEScopy InChI
Affinity DataIC50: 1.07nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometry in presence of 10 uM glycineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50304334(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-tropane | ...)copy SMILEScopy InChI
Affinity DataIC50: 10.2nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)copy SMILEScopy InChI
Affinity DataIC50: 11.5nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50304335(3alpha-(1'-Methyl-2'-Indolecarbonyloxy)-nortropane...)copy SMILEScopy InChI
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50415201(CHEMBL611364)copy SMILEScopy InChI
Affinity DataIC50: 33.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50415204(CHEMBL596443)copy SMILEScopy InChI
Affinity DataIC50: 41.7nMAssay Description:Displacement of [3H]strychnine from GlyR in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 46nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232896(CHEMBL4079657)copy SMILEScopy InChI
Affinity DataIC50: 49nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced currents by whole-ce...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50415205(CHEMBL595797)copy SMILEScopy InChI
Affinity DataIC50: 50.1nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 expressed in HEK293 cells assessed as reduction in glycine-induced whole cell currents ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 51nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 52nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in human tsA201 cells assessed as inhibition of glycine-induced receptor ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50570357(CHEMBL4865147)copy SMILES
Affinity DataIC50: 55nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1 assessed as inhibition of glycine-induced current measured at the later state of compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HH6PV6PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50232890(CHEMBL4102677)copy SMILEScopy InChI
Affinity DataIC50: 56nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 beta expressed in HEK293 cells assessed as inhibition of glycine-induced current at...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1/beta(Homo sapiens (Human))
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50225707(CHEBI:28973 | Strychnine)copy SMILEScopy InChI
Affinity DataIC50: 58nMAssay Description:Antagonist activity at human glycine receptor subunit alpha-1beta expressed in HEK293 cells assessed as reduction in glycine-induced whole cell curre...More data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(RAT)
The German University in Cairo

Curated by ChEMBL
LigandPNGBDBM50415208(CHEMBL608418)copy SMILEScopy InChI
Affinity DataIC50: 58.9nMAssay Description:Displacement of [3H]strychnine from GlyR high affinity site in Wistar rat spinal cord by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DJ5FQJPubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))TBA
LigandPNGBDBM50232889(CHEMBL4103909)copy SMILEScopy InChI
Affinity DataIC50: 59nMAssay Description:Antagonist activity at recombinant human glycine receptor alpha 1 expressed in HEK293 cells assessed as inhibition of glycine-induced current at -50 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QZ2D66PubMed
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