Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Kallikrein-13'
TargetKallikrein-13(Homo sapiens)
Bicycle Therapeutics Limited, Building 900, Babraham Research Campus , Cambridge CB22 3AT , U.K.

Curated by ChEMBL
LigandPNGBDBM50256262(CHEMBL4070056)copy SMILEScopy InChI
Affinity DataKi:  820nMAssay Description:Inhibition of platelet derived growth factor receptor beta phosphorylation in MG63 cells in the presence of human plasmaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JW6PubMed
TargetKallikrein-13(Homo sapiens)
Bicycle Therapeutics Limited, Building 900, Babraham Research Campus , Cambridge CB22 3AT , U.K.

Curated by ChEMBL
LigandPNGBDBM50256261(CHEMBL4059991)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of platelet-derived growth factor receptor beta phosphorylation in MG63 cells in the absence of plasmaMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JW6PubMed
TargetKallikrein-13(Homo sapiens)
Bicycle Therapeutics Limited, Building 900, Babraham Research Campus , Cambridge CB22 3AT , U.K.

Curated by ChEMBL
LigandPNGBDBM50256260(CHEMBL4094403)copy SMILEScopy InChI
Affinity DataKi: >5.00E+4nMAssay Description:Inhibition of recombinant human C-terminal polyHis-tagged KLK13 (1 to 262 residues) expressed in HEK293 cells using fluorogenic Boc-VPR-AMC peptide a...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862JW6PubMed
TargetKallikrein-13(Homo sapiens)
Bicycle Therapeutics Limited, Building 900, Babraham Research Campus , Cambridge CB22 3AT , U.K.

Curated by ChEMBL
LigandPNGBDBM50459539(CHEMBL4206734)copy SMILEScopy InChI
Affinity DataIC50: 500nMAssay Description:Inhibition of KLK13 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q279479BPubMed
TargetKallikrein-13(Homo sapiens)
Bicycle Therapeutics Limited, Building 900, Babraham Research Campus , Cambridge CB22 3AT , U.K.

Curated by ChEMBL
LigandPNGBDBM50459538(CHEMBL4218203)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of KLK13 (unknown origin) expressed in Pichia pastoris pre-incubated for 10 mins before Boc-ValProArg-AMC substrate addition and measured ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q279479BPubMed