Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Muscleblind-like protein 1'
TargetMuscleblind-like protein 1(Homo sapiens)TBA
LigandPNGBDBM15236(3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chr...)copy SMILEScopy InChI
Affinity DataKd:  0.25nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
TargetMuscleblind-like protein 1(Homo sapiens)TBA
LigandPNGBDBM50405589(CHEMBL1710607)copy SMILEScopy InChI
Affinity DataKd:  0.0110nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
TargetMuscleblind-like protein 1(Homo sapiens)TBA
LigandPNGBDBM50408491(CHEMBL4437685)copy SMILEScopy InChI
Affinity DataKd: >2.00E+5nMAssay Description:Antagonist activity at human muscarinic acetylcholine M2 receptor expressed in CHO cells coexpressed with Gqi5 assessed as inhibition of acetylcholin...More data for this Ligand-Target Pair
In DepthDetails
TargetMuscleblind-like protein 1(Homo sapiens)TBA
LigandPNGBDBM50405591(CHEMBL5286270)copy SMILEScopy InChI
Affinity DataKd:  4nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails
TargetMuscleblind-like protein 1(Homo sapiens)TBA
LigandPNGBDBM50405590(CHEMBL5276958)copy SMILEScopy InChI
Affinity DataKd:  93nMAssay Description:In vitro inhibitory activity against beta-2 adrenergic receptor was measured by the inhibition of isoproterenol-induced relaxation of PGF2-alpha cont...More data for this Ligand-Target Pair
In DepthDetails