Compile Data Set for Download or QSAR
Found 15 Enz. Inhib. hit(s) with Target = 'Formyl peptide receptor-related sequence 1'
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50071956(CHEMBL3407845)copy SMILEScopy InChI
Affinity DataEC50:  9.00E+3nMAssay Description:Induction of calcium release in mouse FPR2 receptor-expressed HEK cell by cytosolic-free calcium assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN75KXPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50186957(1-(3-tert-butyl-2-methyl-5-oxo-1-phenyl-2,5-dihydr...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+3nMMore data for this Ligand-Target Pair
In DepthDetails
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097568(CHEMBL3590076)copy SMILEScopy InChI
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097570(CHEMBL3590074)copy SMILEScopy InChI
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097569(CHEMBL3590075)copy SMILEScopy InChI
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097559(CHEMBL3590073)copy SMILEScopy InChI
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097561(CHEMBL3590071)copy SMILEScopy InChI
Affinity DataEC50:  3.90E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097560(CHEMBL3590072)copy SMILEScopy InChI
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097563(CHEMBL3590069)copy SMILEScopy InChI
Affinity DataEC50:  2.50E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097562(CHEMBL3590070)copy SMILEScopy InChI
Affinity DataEC50:  3.80E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097565(CHEMBL3589947)copy SMILEScopy InChI
Affinity DataEC50:  1.70E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097564(CHEMBL3589948)copy SMILEScopy InChI
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097567(CHEMBL3588871)copy SMILEScopy InChI
Affinity DataEC50:  240nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50097566(CHEMBL3589946)copy SMILEScopy InChI
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at FPR2 in BALB/c mouse assessed as stimulation of Ca2+ influx measured every 5 secs for 240 secs by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MS3VHBPubMed
TargetFormyl peptide receptor-related sequence 1(Mus musculus)
Sorbonne Universit£s

Curated by ChEMBL
LigandPNGBDBM50050937((S)-2-[(S)-2-((S)-2-Formylamino-4-methylsulfanyl-b...)copy SMILEScopy InChI
Affinity DataKd: >300nMAssay Description:Binding affinity to mouse FPR2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CN75KXPubMed