TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 0.120nMAssay Description:Inhibition of recombinant C-terminal truncated human SPC6 expressed in drosophila Schneider 2 cells after 1 hr by spectrofluorometryMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 3.60nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 85nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 173nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 188nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 232nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 433nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 492nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 649nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Centre Hospitalier Universitaire Vaudois (CHUV)
Curated by ChEMBL
Affinity DataKi: 806nMAssay Description:Inhibition of human recombinant PC5/6 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair