Compile Data Set for Download or QSAR
Found 7 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha/beta/gamma/delta/epsilon/eta/theta type/Serine/threonine-protein kinase D1/D3'
LigandPNGBDBM50368315(PROSTRATIN)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serumMore data for this Ligand-Target Pair
LigandPNGBDBM50281846((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4VQP
LigandPNGBDBM50281845((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4VQP
LigandPNGBDBM50041403((2R,3R,4R)-2-Hydroxymethyl-5-oxo-4-tetradecyl-tetr...)copy SMILEScopy InChI
Affinity DataKi:  600nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4VQP
LigandPNGBDBM50280454((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-3...)copy SMILEScopy InChI
Affinity DataIC50: 150nMAssay Description:Binding to PKC in 3[H]-PBDU assayMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D50Q4J