Compile Data Set for Download or QSAR
Found 58 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP4'
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50145156(CHEMBL3764816)copy SMILEScopy InChI
Affinity DataIC50: 254nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50145156(CHEMBL3764816)copy SMILEScopy InChI
Affinity DataIC50: 257nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50316226((S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-car...)copy SMILEScopy InChI
Affinity DataIC50: 330nMAssay Description:Inhibition of human v-PARP catalytic domain by trichloroacetic acid precipitation assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DN457MPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 407nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM27566(4-({3-[(4-cyclopropanecarbonylpiperazin-1-yl)carbo...)copy SMILEScopy InChI
Affinity DataIC50: 410nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50306253(1-(2-(pyridin-3-yl)acetyl)-2,3,9,9a-tetrahydro-1H-...)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:Inhibition of VPARPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5N91PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50316226((S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-car...)copy SMILEScopy InChI
Affinity DataIC50: 446nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50316226((S)-2-(4-(piperidin-3-yl)phenyl)-2H-indazole-7-car...)copy SMILEScopy InChI
Affinity DataIC50: 447nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50590271(CHEMBL5198711)copy SMILES
Affinity DataIC50: 500nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KS1PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50306256(1-(3-(pyrazin-2-yl)propanoyl)-2,3,9,9a-tetrahydro-...)copy SMILEScopy InChI
Affinity DataIC50: 660nMAssay Description:Inhibition of VPARPMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GT5N91PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM27497(2-(dimethylamino)-N-(6-oxo-5,6-dihydrophenanthridi...)copy SMILEScopy InChI
Affinity DataIC50: 759nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50590270(CHEMBL5181770)copy SMILES
Affinity DataIC50: 800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KS1PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50590274(CHEMBL5200299)copy SMILES
Affinity DataIC50: 800nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KS1PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataIC50: 832nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50446130(AG-014699 | AG-14447 | RUCAPARIB CAMSYLATE | Rucap...)copy SMILEScopy InChI
Affinity DataIC50: 839nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50590273(CHEMBL5176271)copy SMILES
Affinity DataIC50: 1.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KS1PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50590272(CHEMBL5184065)copy SMILES
Affinity DataIC50: 2.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2H70KS1PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 3.47E+3nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM27135(2-[(2R)-2-methylpyrrolidin-2-yl]-1H-1,3-benzodiazo...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50188594(CHEBI:62878 | CHEMBL1086580)copy SMILEScopy InChI
Affinity DataIC50: 4.37E+3nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50188594(CHEBI:62878 | CHEMBL1086580)copy SMILEScopy InChI
Affinity DataIC50: 4.39E+3nMAssay Description:Inhibition of recombinant human His6-tagged PARP4 ADP-ribosyltransferase domain expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28054VVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50188594(CHEBI:62878 | CHEMBL1086580)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Binding affinity to PARP4 in human Jurkat cell extract after 45 mins by mass spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X350RSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50238428(CHEMBL4087876)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Binding affinity to PARP4 in human Jurkat cell extract after 45 mins by mass spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X350RSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50238425(CHEMBL4064332)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Binding affinity to PARP4 in human Jurkat cell extract after 45 mins by mass spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X350RSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50238416(CHEMBL4087470)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Binding affinity to PARP4 in human Jurkat cell extract after 45 mins by mass spectrometric analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X350RSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50238419(CHEMBL4060134)copy SMILEScopy InChI
Affinity DataIC50: 5.01E+3nMAssay Description:Inhibitory activity against human thymidylate synthase with variable concentration of N5, 10-CH2-H4PteGlu and fixed dUMP (100 uM)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X350RSPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM431646(5-[[(2S)-1-(3-Oxo-3-[4-[5-(trifluoromethyl)pyrimid...)copy SMILES
Affinity DataIC50: 9.20E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5Z03PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50250875(CHEMBL4095003)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR22SXPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50541697(CHEMBL4633637 | US11926614, Example 93)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR22SXPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50541697(CHEMBL4633637 | US11926614, Example 93)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VDHPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50579974(CHEMBL5090849 | US11926614, Example 154 | US202303...)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21R6VDHPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50104285(CHEMBL3593716)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+4nMAssay Description:Inhibition of human ARTD4 (250 to 565) using 500 nM NAD substrate after 2.5 hrs incubationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66NJ2PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4 [250-565](Homo sapiens (Human))
University of Oulu

LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 2.26E+4nMAssay Description:This assay measures the substrate consumption by quantifying the remaining NAD+ through its chemical conversion to a stable fluorescent condensation ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2B56HJ3PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM199181(4-[(4-Carbamoylcyclohexyl)oxy]cyclohexane-1-carbox...)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50104286(CHEMBL3593715)copy SMILEScopy InChI
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of human ARTD4 (250 to 565) using 500 nM NAD substrate after 2.5 hrs incubationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66NJ2PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50234915(CHEMBL4069447)copy SMILEScopy InChI
Affinity DataIC50: 6.46E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9RPPPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50234915(CHEMBL4069447)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9RPPPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50340090(4-methoxybenzamide | CHEMBL449635)copy SMILEScopy InChI
Affinity DataIC50: 6.50E+4nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50234916(CHEMBL4098188)copy SMILEScopy InChI
Affinity DataIC50: 6.90E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9RPPPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50234916(CHEMBL4098188)copy SMILEScopy InChI
Affinity DataIC50: 6.92E+4nMAssay Description:Inhibition of PARP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9RPPPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50104287(CHEMBL3594136)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ARTD4 (250 to 565) using 500 nM NAD substrate after 2.5 hrs incubationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66NJ2PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50104288(CHEMBL3594137)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ARTD4 (250 to 565) using 500 nM NAD substrate after 2.5 hrs incubationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W66NJ2PubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50503853(CHEMBL4545565)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PARP4 BRCT-catalytic domain (1 to 572 residues) assessed as reduction in MARylation of SRPK2 substrate after 60 mins in presence ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HX1GXVPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50468581(CHEMBL4287655)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50452662(CHEMBL4208737)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50468579(CHEMBL4287262)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of N-terminal His-tagged human ARTD4 (250 to 565 residues) expressed in Escherichia coli Rosetta2 (DE3) using TCEP as substrate after 2.5 ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P271SWPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50250875(CHEMBL4095003)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human PARP4 using NAD+ as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8GXGPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50136755(CHEMBL3752386)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ARTD4 by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20003ZDPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50136772(CHEMBL3752492)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human ARTD4 by fluorescence analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20003ZDPubMed
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Health& Science University

Curated by ChEMBL
LigandPNGBDBM50594011(CHEMBL5200521)copy SMILES
Affinity DataIC50: 1.00E+5nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20V8HSSPubMed
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