Compile Data Set for Download or QSAR
Found 82 Enz. Inhib. hit(s) with Target = 'Protein tyrosine phosphatase type IVA 3'
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396097(US10308663, JMS-631-053)copy SMILEScopy InChI
Affinity DataIC50: 18nMAssay Description:The in vitro biochemical evaluation of all compounds was carried out using recombinant human PTP4A3, overexpressed as a His6-tag fusion protein in E....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20867N2US Patent
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396097(US10308663, JMS-631-053)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of recombinant human His6-tagged PRL-3 expressed in Escherichia coli using DiFMUP as substrate incubated for 30 mins by fluorescence based...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50535759(CHEMBL4471843)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant human His-6-tagged PTP4A3 expressed in Escherichia coli assessed as reduction in hydrolysis using DIFMUP as substrate incub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396097(US10308663, JMS-631-053)copy SMILEScopy InChI
Affinity DataIC50: 35nMAssay Description:Inhibition of recombinant human His-6-tagged PTP4A3 expressed in Escherichia coli assessed as reduction in hydrolysis using DIFMUP as substrate incub...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM396097(US10308663, JMS-631-053)copy SMILEScopy InChI
Affinity DataIC50: 84nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571230(CHEMBL4862721)copy SMILES
Affinity DataIC50: 107nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 128nMAssay Description:Inhibition of full length human fusion His6 tagged PRL3 expressed in Escherichia coli using TAMRA-Thr-Ala-Asp-Ile-Tyr(PO3H2)-Glu-NH2 substrate by imm...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z8GPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant human His-6-tagged PTP4A3 expressed in Escherichia coli assessed as increase in polarization using TAMRAThr-Ala-Asp-Ile-Tyr...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 132nMAssay Description:The in vitro biochemical evaluation of all compounds was carried out using recombinant human PTP4A3, overexpressed as a His6-tag fusion protein in E....More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q20867N2US Patent
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571225(CHEMBL4862502)copy SMILES
Affinity DataIC50: 206nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 240nMAssay Description:Inhibition of PRL3 (unknown origin) using DiFMUP as fluorogenic phosphate substrate assessed as DiFMUP dephosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FQ9Z8GPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM45440(4-[5-(4-amidinophenoxy)pentoxy]benzamidine;2-hydro...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of PTP4A3 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50059084(CHEMBL3393171 | US10308663, Thienopyridone (5))copy SMILEScopy InChI
Affinity DataIC50: 460nMAssay Description:Inhibition of full-length human heart His6-tagged PRL-3 expressed in Escherichia coli using DiFMUP as substrate incubated for 35 mins by fluorescence...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50436447(CHEMBL2397162)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of human His6-tagged full length PRL3 assessed as inhibition of DiFMUP dephosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZHJPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184288(5-(2-(2-bromobenzyloxy)-5-bromobenzylidene)-2-thio...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184297(5-(5-(benzo[b]thiophen-3-yl)-2-(benzyloxy)benzylid...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184288(5-(2-(2-bromobenzyloxy)-5-bromobenzylidene)-2-thio...)copy SMILEScopy InChI
Affinity DataIC50: 900nMAssay Description:Inhibition of PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8SHKPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184288(5-(2-(2-bromobenzyloxy)-5-bromobenzylidene)-2-thio...)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human His6-tagged full length PRL3 assessed as inhibition of DiFMUP dephosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2QR4ZHJPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571229(CHEMBL4852178)copy SMILES
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184287(5-(5-(benzofuran-3-yl)-2-(benzyloxy)benzylidene)-2...)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184285(5-(2-(4-bromobenzyloxy)benzylidene)-2-thioxothiazo...)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184298(5-(4-Benzyloxy-biphenyl-3-ylmethylene)-2-thioxo-th...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184296(5-((3-(2-chloro-6-fluorobenzyloxy)naphthalen-2-yl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184293(5-[1-[3-(biphenyl-4-ylmethoxy)-naphthalen-2-yl]-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571226(CHEMBL4864481)copy SMILES
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184291(5-((3-(benzyloxy)naphthalen-2-yl)methylene)-2-thio...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184290(5-(2-(2-chlorobenzyloxy)-5-bromobenzylidene)-2-thi...)copy SMILEScopy InChI
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184294(5-(2-(benzyloxy)-5-bromobenzylidene)-2-thioxothiaz...)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184292(5-((3-(3,5-dimethoxybenzyloxy)naphthalen-2-yl)meth...)copy SMILEScopy InChI
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)copy SMILEScopy InChI
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of PRL3 after 1 hr by DiFMUP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K074QMPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184289(5-[1-(4-benzyloxy-4'-dimethylamino-biphenyl-3-yl)-...)copy SMILEScopy InChI
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184286(5-(2-(benzyloxy)-5-bromobenzyl)-2-thioxothiazolidi...)copy SMILEScopy InChI
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50312665(CHEMBL1088572 | Sodium 2-(2-Fluorophenyl)-6,7-meth...)copy SMILEScopy InChI
Affinity DataIC50: 4.93E+3nMAssay Description:Inhibition of human PTP4A3 by enzyme assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XG9R8XPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571227(CHEMBL4854258)copy SMILES
Affinity DataIC50: 4.98E+3nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50571228(CHEMBL4856668)copy SMILES
Affinity DataIC50: 6.59E+3nMAssay Description:Inhibition of recombinant human PTP4A3More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23X8BDDPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50184295((Z)-5-(5-bromo-2-hydroxybenzylidene)-2-thioxothiaz...)copy SMILEScopy InChI
Affinity DataIC50: 9.50E+3nMAssay Description:Inhibition of human recombinant PRL-3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB746WPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50391711(CHEMBL2146958)copy SMILEScopy InChI
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of PRL3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2QDCPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237949(2-(5-((4-oxo-2-thioxothiazolidin-5-ylidene)methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of recombinant human PTP4A3 expressed in Escherichia coli BL21 (DE3) assessed as reduction in hydrolysis using DIFMUP as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237949(2-(5-((4-oxo-2-thioxothiazolidin-5-ylidene)methyl)...)copy SMILEScopy InChI
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human PRL3 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1X08PubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50569365(CHEMBL4867742)copy SMILES
Affinity DataIC50: 1.52E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237952(3-(2-((1-(3-chlorophenyl)-2,5-dioxoimidazolidin-4-...)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of human PRL3 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1X08PubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50535760(CHEMBL4466901)copy SMILEScopy InChI
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibition of recombinant human PTP4A3 expressed in Escherichia coli BL21 (DE3) assessed as reduction in hydrolysis using DIFMUP as substrate incubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237948((E)-2-(2-(5-(4-chlorophenyl)furan-2-yl)vinyl)-6-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of human PRL3 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1X08PubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237948((E)-2-(2-(5-(4-chlorophenyl)furan-2-yl)vinyl)-6-me...)copy SMILEScopy InChI
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of recombinant human PTP4A3 expressed in Escherichia coli BL21 (DE3) assessed as reduction in hydrolysis using DIFMUP as substrate incubat...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VH5SBFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50569366(CHEMBL4858539)copy SMILES
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50323199(5,7-dihydroxy-8-(5-(5-hydroxy-7-methoxy-4-oxo-4H-c...)copy SMILEScopy InChI
Affinity DataIC50: 2.58E+4nMAssay Description:Inhibition of human brain PRL-3 (1 to 168 residues) expressed in Escherichia coli BL21(DE3) cells using DiFMUP as substrate incubated for 1 hr by flu...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50569362(CHEMBL1699070)copy SMILES
Affinity DataIC50: 2.60E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50569367(CHEMBL4850661)copy SMILES
Affinity DataIC50: 2.67E+4nMAssay Description:Inhibition of PRL-3 (unknown origin) using DiFMUP as substrate incubated for 1 hrMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2NK3JSFPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50391714(CHEMBL2146957)copy SMILEScopy InChI
Affinity DataIC50: 2.76E+4nMAssay Description:Inhibition of PRL3More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2QDCPubMed
TargetProtein tyrosine phosphatase type IVA 3(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals Inc.

LigandPNGBDBM50237950(3-benzylsulfanyl-6-[1-(4-hydroxy-3-methoxy-phenyl)...)copy SMILEScopy InChI
Affinity DataIC50: 2.77E+4nMAssay Description:Inhibition of human PRL3 expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q1X08PubMed
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