Compile Data Set for Download or QSAR
Found 11 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor gamma [183-417]'
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31889(BMS 961 | BMS270394 | BMS961)copy SMILEScopy InChI
Affinity DataKi:  1.5nM ΔG°:  -46.8kJ/molepH: 8.0 T: 2°CAssay Description:Competitive assay were perform with 5nM tritiated all-trans retinoic acid (t-RA; 5nM) with or without 100-fold excess of non-radioactive t-RA (500nM)...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31884(BMS184394-S | CHEMBL81273)copy SMILEScopy InChI
Affinity DataKd:  816nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31885(BMS184394 | CHEMBL82089)copy SMILEScopy InChI
Affinity DataKd:  64nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31886(CD564 | CHEMBL309282)copy SMILEScopy InChI
Affinity DataKd:  3nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31887(BMS181156 | Ch 80)copy SMILEScopy InChI
Affinity DataKd:  0.600nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31889(BMS 961 | BMS270394 | BMS961)copy SMILEScopy InChI
Affinity DataKd:  528nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31890(BMS270395)copy SMILEScopy InChI
Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31883(9-cis-retinoic acid (9cRA) | ALL-TRANS-RETINOIC AC...)copy SMILEScopy InChI
Affinity DataKd:  0.200nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8QHRPubMedMMDB
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31892(9-cis retinoic acid | 9C-RA | CHEMBL705 | Panretin...)copy SMILEScopy InChI
Affinity DataKd:  0.800nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31882(BMS184394-R | CHEMBL80992)copy SMILEScopy InChI
Affinity DataKd:  75nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8QHRPubMed
TargetRetinoic acid receptor gamma [183-417](Homo sapiens (Human))
Institut de Génétique et de Biologie Moléculaire et Cellulaire (IGBMC)

LigandPNGBDBM31888(CD666)copy SMILEScopy InChI
Affinity DataKd:  68nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8QHRPubMed