Compile Data Set for Download or QSAR
Found 10 Enz. Inhib. hit(s) with Target = 'Segment polarity protein dishevelled homolog DVL-3'
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373848(CHEMBL255779)copy SMILEScopy InChI
Affinity DataIC50: 2.30E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373844(CHEMBL272948)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373845(CHEMBL402939)copy SMILEScopy InChI
Affinity DataIC50: 9.20E+4nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373851(CHEMBL256431)copy SMILEScopy InChI
Affinity DataIC50: 1.60E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373846(CHEMBL401537)copy SMILEScopy InChI
Affinity DataIC50: 2.91E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373847(CHEMBL256605)copy SMILEScopy InChI
Affinity DataIC50: 3.09E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373843(CHEMBL410400)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373849(CHEMBL255988)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50373850(CHEMBL404331)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed
TargetSegment polarity protein dishevelled homolog DVL-3(Homo sapiens (Human))
St. Jude Children's Research Hospital

Curated by ChEMBL
LigandPNGBDBM50231890(2-((2-carboxyethyl)carbamoyl)-6-methyl-3-phenethyl...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMAssay Description:Antagonist activity at human Dvl3 assessed as inhibition of interaction between Dvl3 PDZ domain and Fz7 PDZ domain by alphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25D8SPTPubMed