Found 11 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 9 subunit alpha/subunit beta-1' TargetSodium channel protein type 9 subunit alpha/subunit beta-1/subunit beta-2(Mus musculus)
Daiichi Sankyo Co., Ltd.
Curated by ChEMBL
Daiichi Sankyo Co., Ltd.
Curated by ChEMBL
Affinity DataIC50: 0.550nMAssay Description:Inhibition of mouse NaV1.7/beta1/beta2 expressed in HEK293A cells by Ionworks high-throughput electrophysiology methodMore data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 258nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 258nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 297nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 297nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 510nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 625nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 625nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 664nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
TargetSodium channel protein type 9 subunit alpha/subunit beta-1(Homo sapiens (Human))
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Xenon Pharmaceuticals Inc.
Curated by ChEMBL
Affinity DataIC50: 664nMAssay Description:Inhibition of recombinant human full length Nav1.7 co-expressed with human SCN1B in HEK293 cells measured after 20 mins at -60 mV holding potential b...More data for this Ligand-Target Pair
