Compile Data Set for Download or QSAR
Found 5 Enz. Inhib. hit(s) with Target = 'Disintegrin and metalloproteinase domain-containing protein 12'
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50062351((R)-N*4*-Hydroxy-N*1*-[(S)-2-(1H-indol-3-yl)-1-met...)copy SMILEScopy InChI
Affinity DataIC50: 5.93nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156477(CHEMBL366034 | {3-(3-Bromo-phenyl)-2-[(furan-2-car...)copy SMILEScopy InChI
Affinity DataIC50: 16.7nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156475(2-[2-[(5-Bromo-furan-2-carbonyl)-amino]-3-(4-bromo...)copy SMILEScopy InChI
Affinity DataIC50: 24.8nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156476(2-[2-Benzoylamino-3-(2-fluoro-phenyl)-acryloylamin...)copy SMILEScopy InChI
Affinity DataIC50: 40.5nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed
TargetDisintegrin and metalloproteinase domain-containing protein 12(Homo sapiens (Human))
Department of Life Science and National Research Laboratory of Proteolysis

Curated by ChEMBL
LigandPNGBDBM50156478(2-{2-[(Furan-2-carbonyl)-amino]-3-furan-2-yl-acryl...)copy SMILEScopy InChI
Affinity DataIC50: 42.3nMAssay Description:Inhibition of A disintegrin and metalloproteinase domain 12 (ADAM12) binding in cell based assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z94DHPubMed