Compile Data Set for Download or QSAR
Found 36 Enz. Inhib. hit(s) with Target = 'Protein ADM2'
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570409(CHEMBL4857810)copy SMILES
Affinity DataIC50: 0.631nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570410(CHEMBL4851152)copy SMILES
Affinity DataIC50: 1nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570411(CHEMBL4877585)copy SMILES
Affinity DataIC50: 1.60nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570413(CHEMBL4850259)copy SMILES
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570396(CHEMBL4871934)copy SMILES
Affinity DataIC50: 6.30nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570397(CHEMBL4852669)copy SMILES
Affinity DataIC50: 7.90nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50246690(Ac-WVTHRLAGLLSRSGGVVRKNFVPTDVGPFAF-NH2 | CHEMBL503...)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570401(CHEMBL4879142)copy SMILES
Affinity DataIC50: 32nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570400(CHEMBL4876643)copy SMILES
Affinity DataIC50: 79nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570402(CHEMBL4856402)copy SMILES
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570408(CHEMBL4873687)copy SMILES
Affinity DataIC50: 100nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50246693(Ac-WVTH[Cit]LAGLLS[Cit]SGGVVRKNFVPTDVGPFAF-NH2 | C...)copy SMILEScopy InChI
Affinity DataIC50: 108nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570404(CHEMBL4850583)copy SMILES
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570398(CHEMBL4861626)copy SMILES
Affinity DataIC50: 126nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570388(CHEMBL4858139)copy SMILES
Affinity DataIC50: 200nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50000743(CHEMBL525571 | [Thr-His-Arg-Leu-Ala-Gly-Leu-Leu-Se...)copy SMILEScopy InChI
Affinity DataIC50: 266nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570394(CHEMBL4866548)copy SMILES
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570395(CHEMBL4866915)copy SMILES
Affinity DataIC50: 316nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50246697(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGPFAF-NH...)copy SMILEScopy InChI
Affinity DataIC50: 318nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50246708(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[1-Nal...)copy SMILEScopy InChI
Affinity DataIC50: 375nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50246709(Ac-WVTH[Cit]LAGLLS[Cit]SGGVV[hArg]KNFVPTDVGP[2-Nal...)copy SMILEScopy InChI
Affinity DataIC50: 418nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50025073(CHEMBL2372187)copy SMILEScopy InChI
Affinity DataIC50: 496nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570406(CHEMBL4862324)copy SMILES
Affinity DataIC50: 501nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570412(CHEMBL4853766)copy SMILES
Affinity DataIC50: 794nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570390(CHEMBL4851106)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570405(CHEMBL4874859)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570393(CHEMBL4878394)copy SMILES
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570386(CHEMBL4864804)copy SMILES
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570403(CHEMBL4874651)copy SMILES
Affinity DataIC50: 1.26E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570407(CHEMBL4865654)copy SMILES
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50025076(CHEMBL2372194)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human adrenomedullin 2 receptor expressed in CHO cells assessed as effect on cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P26Z0CPubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570399(CHEMBL4846989)copy SMILES
Affinity DataIC50: 3.16E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570392(CHEMBL4870543)copy SMILES
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570389(CHEMBL4867733)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570387(CHEMBL4853613)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed
TargetProtein ADM2(Homo sapiens (Human))TBA
LigandPNGBDBM50570391(CHEMBL4876213)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at human AM2 expressed in 1321N1 cells assessed as inhibition of forskolin-induced cAMP accumulation preincubated for 30 mins fol...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2474FM7PubMed