Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Antithrombin-III/Prothrombin'
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264613(US9718760, C157)copy SMILEScopy InChI
Affinity DataIC50: 4.44E+4nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264597(US9718760, C152)copy SMILEScopy InChI
Affinity DataIC50: 8.70E+4nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264614(US9718760, C158)copy SMILEScopy InChI
Affinity DataIC50: 5.47E+5nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264648(US9718760, C161)copy SMILEScopy InChI
Affinity DataIC50: 1.67E+6nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264598(US9718760, C155)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+6nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent
TargetAntithrombin-III/Prothrombin(Homo sapiens (Human))
THE REGENTS OF THE UNIVERSITY OF MICHIGAN; EASTERN MICHIGAN UNIVERSITY

US Patent
LigandPNGBDBM264627(US9718760, C160)copy SMILEScopy InChI
Affinity DataIC50: 2.33E+6nMT: 2°CAssay Description:PAI-1 inhibitor compounds were dissolved in DMSO to a final concentration of (10-50 mM), depending upon solubility. Compounds were then diluted in ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2K939HKUS Patent