Compile Data Set for Download or QSAR
Found 15 Enz. Inhib. hit(s) with Target = 'Accessory gene regulator protein A'
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020375(CHEMBL3289785)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50499936(CHEMBL3742171)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868BFPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50499937(CHEBI:67522 | Turnagainolide A)copy SMILEScopy InChI
Affinity DataIC50: 800nMAssay Description:Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868BFPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50499939(CHEMBL3740058)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868BFPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50499938(CHEMBL3741390)copy SMILEScopy InChI
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of agr-mediated quorum sensing in Staphylococcus aureus after 5 hrs by luminescence analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20868BFPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of Staphylococcus aureus RN6390B Agr-mediated RNA3 promoter activation measured up to 6 hrs by Northern blot analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BV7J0MPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020376(CHEBI:81348 | CHEMBL290932)copy SMILEScopy InChI
Affinity DataIC50: 8.10E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020377(CHEMBL3289786)copy SMILEScopy InChI
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM11318(1,3,8-trihydroxy-6-methyl-9,10-dihydroanthracene-9...)copy SMILEScopy InChI
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020378(CHEMBL3289787)copy SMILEScopy InChI
Affinity DataIC50: 1.98E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020379(CHEMBL3289788)copy SMILEScopy InChI
Affinity DataIC50: 2.65E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020380(CHEMBL3289789)copy SMILEScopy InChI
Affinity DataIC50: 3.01E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM115127(4,5,7-trihydroxy-9,10-diketo-anthracene-2-carboxyl...)copy SMILEScopy InChI
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50312649(6-chloro-4,5,7-trihydroxy-9,10-dioxo-9,10-dihydroa...)copy SMILEScopy InChI
Affinity DataIC50: 3.78E+4nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed
TargetAccessory gene regulator protein A(Staphylococcus aureus)
University of North Carolina at Greensboro

Curated by ChEMBL
LigandPNGBDBM50020389(CHEMBL3289790)copy SMILEScopy InChI
Affinity DataIC50: 1.20E+5nMAssay Description:Inhibition of AGR quorum sensing system in methicillin-resistant Staphylococcus aureus AH2759 incubated for 15 hrs by P3-LUX reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q21V5GJDPubMed