Compile Data Set for Download or QSAR
Found 58 Enz. Inhib. hit(s) with Target = 'Acid-sensing ion channel 1'
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50096642(CHEMBL3577296)copy SMILEScopy InChI
Affinity DataIC50: 27nMpH: 6.7Assay Description:Inhibition of human ASIC1a endogenously expressed in HEK293 cells clamped at -100 mV gated ionic current at pH 6.7 by standard whole cell patch clamp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NTKPubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50348098(CHEMBL1800430)copy SMILEScopy InChI
Affinity DataIC50: 224nMAssay Description:Inhibition of ASIC1aMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DZ08P8PubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408492(CHEMBL5269133)copy SMILEScopy InChI
Affinity DataIC50: 407nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408498(CHEMBL5270983)copy SMILEScopy InChI
Affinity DataIC50: 518nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408502(CHEMBL5289168)copy SMILEScopy InChI
Affinity DataIC50: 729nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408500(CHEMBL5278611)copy SMILEScopy InChI
Affinity DataIC50: 972nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408497(CHEMBL5287933)copy SMILEScopy InChI
Affinity DataIC50: 1.42E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408496(CHEMBL5291421)copy SMILEScopy InChI
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408493(CHEMBL5285672)copy SMILEScopy InChI
Affinity DataIC50: 1.99E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50157090(6-(2-(1-isopropyl-2-methyl-1,2,3,4-tetrahydroisoqu...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of ASIC1a in rat dorsal root ganglion neurons assessed as reduction in peak current preincubated for 120 secs followed by acid medium stim...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2PZ5CBDPubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408495(CHEMBL5267130)copy SMILEScopy InChI
Affinity DataIC50: 2.59E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408499(CHEMBL5276647)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408494(CHEMBL5267106)copy SMILEScopy InChI
Affinity DataIC50: 3.14E+3nMAssay Description:Antagonist activity at human muscarinic acetylcholine M1 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobi...More data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50096642(CHEMBL3577296)copy SMILEScopy InChI
Affinity DataIC50: 7.34E+3nMpH: 5.0Assay Description:Inhibition of human ASIC1a endogenously expressed in HEK293 cells clamped at -100 mV gated ionic current at pH 5.0 by standard whole cell patch clamp...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FT8NTKPubMed
TargetAcid-sensing ion channel 1(Homo sapiens (Human))
Bogomoletz Institute of Physiology of NAS Ukraine

Curated by ChEMBL
LigandPNGBDBM50408501(CHEMBL5283083)copy SMILEScopy InChI
Affinity DataIC50: 9.54E+3nMAssay Description:Antagonist activity at AT1 receptor in rat aortaMore data for this Ligand-Target Pair
In DepthDetails
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510042(CHEMBL4593172)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510052(CHEMBL4446500)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510049(CHEMBL4590631)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510057(CHEMBL4538655)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510055(CHEMBL4440787)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510050(CHEMBL4463485)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1/2(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510034(CHEMBL4593063)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.25-stimulated mouse ASIC1a/2a heterodimer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510034(CHEMBL4593063)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510035(CHEMBL4528810)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510038(CHEMBL4518161)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510039(CHEMBL4456021)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510040(CHEMBL4469611)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510041(CHEMBL4476781)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510056(CHEMBL4450681)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510043(CHEMBL4524195)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510044(CHEMBL4462808)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510045(CHEMBL4587871)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510046(CHEMBL4440380)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510047(CHEMBL4517411)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510048(CHEMBL4442568)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510037(CHEMBL4463769)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510036(CHEMBL4555958)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510054(CHEMBL4445209)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510053(CHEMBL4591499)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50510051(CHEMBL4527919)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM16173(3,5-diamino-6-chloro-N-(diaminomethylene)pyrazinam...)copy SMILEScopy InChI
Affinity DataIC50: 3.02E+4nMAssay Description:Inhibition of ASIC1 in Sprague-Dawley rat articular chondrocytes assessed as decrease in acid-induced intracellular calcium level by Fluo-3AM dye bas...More data for this Ligand-Target Pair
TargetAcid-sensing ion channel 1(Mus musculus)
Promidis

Curated by ChEMBL
LigandPNGBDBM50000999(CHEBI:81724 | DIMINAZENE)copy SMILEScopy InChI
Affinity DataIC50: 5.69E+4nMAssay Description:Inhibition of pH 6.6-stimulated mouse ASIC1a homomer expressed in CHOK1 cells assessed as reduction in channel activation by VSD fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RB77Z0PubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes at pH 6.4 by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)copy SMILEScopy InChI
Affinity DataIC50: 1.35E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes at pH 6.9 by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50074922((+-)-2-fluoro-alpha-methyl-4-biphenylacetic acid |...)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes assessed as inhibition of pH 6.7-gated currents by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50250133(Butibufen)copy SMILEScopy InChI
Affinity DataIC50: 1.82E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes assessed as inhibition of pH 6.7-gated currents by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50169044((-)-ibuprofen | (2R)-2-(4-isobutylphenyl)propanoic...)copy SMILEScopy InChI
Affinity DataIC50: 2.88E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes assessed as inhibition of pH 6.7-gated currents by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes at pH 6.7 by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes at pH 6.7 by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
TargetAcid-sensing ion channel 1(Rattus norvegicus)
Anhui Medical University

Curated by ChEMBL
LigandPNGBDBM50009859((+-)-2-(p-isobutylphenyl)propionic acid | (+-)-alp...)copy SMILEScopy InChI
Affinity DataIC50: 2.95E+5nMAssay Description:Inhibition of rat ASIC1a receptor expressed in xenopus lavies oocytes assessed as inhibition of pH 6.7-gated currents by two electrode voltage clampMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N58PSVPubMed
Displayed 1 to 50 (of 58 total ) | Next | Last >>
Jump to: