Compile Data Set for Download or QSAR
Found 47 Enz. Inhib. hit(s) with Target = 'Apoptosis regulator BAX'
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50570680(CHEMBL4868313)copy SMILES
Affinity DataKi:  43nMAssay Description:Displacement of Bak BH3 domain peptide from human Bax by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2P272X3PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataKi:  800nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078029(CHEMBL3417409)copy SMILEScopy InChI
Affinity DataKi:  1.00E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078027(CHEMBL3417407)copy SMILEScopy InChI
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078026(CHEMBL3417406)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078028(CHEMBL3417408)copy SMILEScopy InChI
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078024(CHEMBL3417404)copy SMILEScopy InChI
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078030(CHEMBL3417410)copy SMILEScopy InChI
Affinity DataKi:  2.50E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078023(CHEMBL3417403)copy SMILEScopy InChI
Affinity DataKi:  9.10E+3nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078018(CHEMBL3417398)copy SMILEScopy InChI
Affinity DataKi:  1.26E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078017(CHEMBL3417397)copy SMILEScopy InChI
Affinity DataKi:  1.29E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078016(CHEMBL3417396)copy SMILEScopy InChI
Affinity DataKi:  1.35E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078019(CHEMBL3417399)copy SMILEScopy InChI
Affinity DataKi:  1.58E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078025(CHEMBL3417405)copy SMILEScopy InChI
Affinity DataKi:  3.09E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078020(CHEMBL3417400)copy SMILEScopy InChI
Affinity DataKi:  6.31E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078021(CHEMBL3417401)copy SMILEScopy InChI
Affinity DataKi:  8.51E+4nMAssay Description:Displacement of FITC-BIM from recombinant N-terminal GST-tagged human BAX expressed in Escherichia coli after 30 mins by fluorescence polarization as...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50516397(CHEMBL4579601)copy SMILEScopy InChI
Affinity DataIC50: 43nMAssay Description:Displacement of fluorescent Bak BH3 peptide domain from human recombinant Bax by competition fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZP49F8PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610526(CHEMBL5282360)copy SMILES
Affinity DataIC50: 250nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547480(CHEMBL4790235)copy SMILES
Affinity DataIC50: 250nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50540081(CHEMBL4438921)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+3nMAssay Description:Activation of Bax in human SMMC7721 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2ZP7PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547494(CHEMBL4783072)copy SMILES
Affinity DataIC50: 3.30E+3nMAssay Description:Activation of BAX (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610527(CHEMBL5266955)copy SMILES
Affinity DataIC50: 3.30E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610529(CHEMBL5278460)copy SMILES
Affinity DataIC50: 4.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610530(CHEMBL5271207)copy SMILES
Affinity DataIC50: 6.00E+3nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547484(CHEMBL4780328)copy SMILES
Affinity DataEC50:  809nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547486(CHEMBL4790418)copy SMILES
Affinity DataEC50:  2.22E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547487(CHEMBL4761391)copy SMILES
Affinity DataEC50:  725nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547488(CHEMBL4797324)copy SMILES
Affinity DataEC50:  967nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547489(CHEMBL4758680)copy SMILES
Affinity DataEC50:  925nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547490(CHEMBL4756429)copy SMILES
Affinity DataEC50:  856nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547491(CHEMBL4784916)copy SMILES
Affinity DataEC50:  532nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547492(CHEMBL4779693)copy SMILES
Affinity DataEC50:  538nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547493(CHEMBL4776616)copy SMILES
Affinity DataEC50:  992nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547480(CHEMBL4790235)copy SMILES
Affinity DataEC50:  278nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)copy SMILEScopy InChI
Affinity DataEC50: >1.00E+4nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547483(CHEMBL4778142)copy SMILES
Affinity DataEC50:  719nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547482(CHEMBL4754714)copy SMILES
Affinity DataEC50:  874nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547481(CHEMBL4777011)copy SMILES
Affinity DataEC50:  704nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610525(CHEMBL4578793)copy SMILES
Affinity DataKd:  255nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM398051(US10322118, Entry 9)copy SMILEScopy InChI
Affinity DataKd:  3.70E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078022(CHEMBL3417402)copy SMILEScopy InChI
Affinity DataEC50:  700nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50078015(CHEMBL3417395)copy SMILEScopy InChI
Affinity DataEC50:  8.20E+3nMAssay Description:Activation of Bax in human HuH7 cells assessed as inhibition of mitochondrial accumulation of fluorescent probe Mitotracker Red after 12 to 72 hrs by...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2X35055PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50610528(CHEMBL5289201)copy SMILES
Affinity DataKd:  1.50E+4nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM196140(US9211296, Table 7, Compd: 13)copy SMILEScopy InChI
Affinity DataKd:  1.50E+4nMMore data for this Ligand-Target Pair
In DepthDetails
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547485(CHEMBL4753330)copy SMILES
Affinity DataEC50:  1.14E+3nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed
TargetApoptosis regulator BAX(Homo sapiens (Human))TBA
LigandPNGBDBM50547479(CHEMBL4794290)copy SMILES
Affinity DataEC50:  393nMAssay Description:Binding affinity to recombinant human full length His-tagged BAX expressed in Escherichia coli BL21 (DE3) cells preincubated for 30 min followed by F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2N301J4PubMed