Compile Data Set for Download or QSAR
Found 3 Enz. Inhib. hit(s) with Target = 'Bromodomain-containing protein 3 [306-416]'
TargetBromodomain-containing protein 3 [306-416](Homo sapiens (Human))
Dana-Farber Cancer Institute

LigandPNGBDBM205431((6S+2S)-PEG1 (7))copy SMILEScopy InChI
Affinity DataKi:  0.00270nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ31HWPubMed
TargetBromodomain-containing protein 3 [306-416](Homo sapiens (Human))
Dana-Farber Cancer Institute

LigandPNGBDBM205453(MTI (35))copy SMILEScopy InChI
Affinity DataKi:  0.0700nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ31HWPubMed
TargetBromodomain-containing protein 3 [306-416](Homo sapiens (Human))
Dana-Farber Cancer Institute

LigandPNGBDBM205429( (R)-JQ1 (3) | US10407441, Compound (R)-JQ1 | US10...)copy SMILEScopy InChI
Affinity DataKd:  19nMAssay Description:Refer to DiscoverXMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VQ31HWPubMed