Compile Data Set for Download or QSAR
Found 12 Enz. Inhib. hit(s) with Target = 'Cyclin-K/Cyclin-dependent kinase 9'
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525738(US11174252, Compound 33)copy SMILES
Affinity DataIC50: 2nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525743(US11174252, Compound 38)copy SMILES
Affinity DataIC50: 2nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525729(US11174252, Compound 24)copy SMILES
Affinity DataIC50: 4nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525750(US11174252, Compound 437)copy SMILES
Affinity DataIC50: 4nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525730(US11174252, Compound 25)copy SMILES
Affinity DataIC50: 5nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50059889((staurosporine)3-methoxy-2-methyl-4-methylamino-(2...)copy SMILEScopy InChI
Affinity DataIC50: 13nMAssay Description:Inhibition of CDK9/Cyclin K (unknown origin)-mediated phosphorylation of peptide substrate incubated for 15 mins prior to substrate addition measured...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25T3MV7PubMed
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525755(US11174252, Compound 442)copy SMILES
Affinity DataIC50: 41nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525749(US11174252, Compound 436)copy SMILES
Affinity DataIC50: 73nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525760(US11174252, Compound 447)copy SMILES
Affinity DataIC50: 243nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM525759(US11174252, Compound 446)copy SMILES
Affinity DataIC50: 280nMAssay Description:CDK9 (cyclin K): IC50 values of compounds against CDK9 (cyclin K) were determined by LanthaScreen™ Eu Kinase Binding Assay at Invitrogen Life Te...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q27D2Z99US Patent
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50263013(CHEMBL4079206)copy SMILEScopy InChI
Affinity DataIC50: 412nMAssay Description:Inhibition of CDK9/cyclin K (unknown origin) after 30 mins in presence of [33P]-gamma-ATP by filter binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DV1NC4PubMed
TargetCyclin-K/Cyclin-dependent kinase 9(Homo sapiens (Human))TBA
LigandPNGBDBM50526803(CHEMBL4434871 | US10870651, Compound 101)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+3nMAssay Description:Compounds of the invention were assayed for activity against a variety of different kinases.More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QZ2F2TUS Patent