Compile Data Set for Download or QSAR
Found 6 Enz. Inhib. hit(s) with Target = 'Proprotein convertase subtilisin/kexin type 4'
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50270054(CHEMBL502642 | TPRARRRKKRT)copy SMILEScopy InChI
Affinity DataKi:  441nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50270060(CHEMBL455792 | TPQRARRRKKRT)copy SMILEScopy InChI
Affinity DataKi:  515nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50269901(CHEMBL525748 | TPRARRRKKRI)copy SMILEScopy InChI
Affinity DataKi:  562nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50270069(CHEMBL499438 | TPQRARRRKKRY)copy SMILEScopy InChI
Affinity DataKi:  624nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50270068(CHEMBL500184 | TPQRARRRKKRF)copy SMILEScopy InChI
Affinity DataKi:  772nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed
TargetProprotein convertase subtilisin/kexin type 4(Homo sapiens (Human))
Institute for Medical Research

Curated by ChEMBL
LigandPNGBDBM50270067(CHEMBL503520 | TPQRARRRKKRW)copy SMILEScopy InChI
Affinity DataKi:  952nMAssay Description:Inhibition of human recombinant PC4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavageMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2057FPBPubMed