Compile Data Set for Download or QSAR
Found 56 Enz. Inhib. hit(s) with Target = 'Tau-tubulin kinase 2'
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50609151(CHEMBL5283456)copy SMILES
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50609159(CHEMBL5280210)copy SMILES
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602886(CHEMBL5182036)copy SMILES
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50609146(CHEMBL5273263)copy SMILES
Affinity DataIC50: 13nMMore data for this Ligand-Target Pair
Ligand InfoPDB
In DepthDetails
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602885(CHEMBL5193906)copy SMILES
Affinity DataIC50: 170nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50506660(CHEMBL4528881)copy SMILEScopy InChI
Affinity DataIC50: 170nMAssay Description:Inhibition of TTBK2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2V98CC0PubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602917(CHEMBL5200069)copy SMILES
Affinity DataIC50: 490nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602903(CHEMBL5198544)copy SMILES
Affinity DataIC50: 850nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602907(CHEMBL5193488)copy SMILES
Affinity DataIC50: 970nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602926(CHEMBL5200160 | US11814388, Compound 9)copy SMILES
Affinity DataIC50: 1.21E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602909(CHEMBL5197789)copy SMILES
Affinity DataIC50: 1.21E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602910(CHEMBL5209196)copy SMILES
Affinity DataIC50: 1.24E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602900(CHEMBL5185704 | US11814388, Compound 3)copy SMILES
Affinity DataIC50: 1.32E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602899(CHEMBL5207783)copy SMILES
Affinity DataIC50: 1.68E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602933(CHEMBL5178462)copy SMILES
Affinity DataIC50: 1.75E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602931(CHEMBL5197012)copy SMILES
Affinity DataIC50: 2.03E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602906(CHEMBL5187459)copy SMILES
Affinity DataIC50: 2.14E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602932(CHEMBL5178965)copy SMILES
Affinity DataIC50: 2.61E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602920(CHEMBL5187125)copy SMILES
Affinity DataIC50: 2.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602930(CHEMBL5181249)copy SMILES
Affinity DataIC50: 2.75E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602929(CHEMBL5193034)copy SMILES
Affinity DataIC50: 2.87E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602905(CHEMBL5208565)copy SMILES
Affinity DataIC50: 3.02E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602922(CHEMBL5184336)copy SMILES
Affinity DataIC50: 3.05E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602923(CHEMBL5178871)copy SMILES
Affinity DataIC50: 3.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50506661(CHEMBL4517951)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602904(CHEMBL5204869)copy SMILES
Affinity DataIC50: 4.22E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602921(CHEMBL5180098)copy SMILES
Affinity DataIC50: 4.49E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602911(CHEMBL5171328)copy SMILES
Affinity DataIC50: 4.90E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602925(CHEMBL5188513)copy SMILES
Affinity DataIC50: 4.94E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602928(CHEMBL5209161)copy SMILES
Affinity DataIC50: 5.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602898(CHEMBL5171736)copy SMILES
Affinity DataIC50: 5.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602919(CHEMBL5169390)copy SMILES
Affinity DataIC50: 5.72E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602934(CHEMBL5206548)copy SMILES
Affinity DataIC50: 6.05E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602913(CHEMBL5207918)copy SMILES
Affinity DataIC50: 6.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602888(CHEMBL5204443)copy SMILES
Affinity DataIC50: 6.70E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602916(CHEMBL5196033)copy SMILES
Affinity DataIC50: 6.79E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602889(CHEMBL5186693)copy SMILES
Affinity DataIC50: 7.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602896(CHEMBL5182006)copy SMILES
Affinity DataIC50: 7.58E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602901(CHEMBL5202436)copy SMILES
Affinity DataIC50: 8.40E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602912(CHEMBL5179559)copy SMILES
Affinity DataIC50: 8.79E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50328192(CHEMBL1257781 | N-(4-(Trifluoromethoxy)phenyl)-7H-...)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+3nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602897(CHEMBL5209114)copy SMILES
Affinity DataIC50: 9.30E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50044784(CHEBI:79090 | SB-202190 | US10865384, Compound SB2...)copy SMILEScopy InChI
Affinity DataIC50: 9.34E+3nMAssay Description:Inhibition of human TTBK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2W380MTPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602918(CHEMBL5193008)copy SMILES
Affinity DataIC50: 9.54E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50519662(CHEMBL4438748)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human TTBK2 (1 to331 residues) using casein as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2MC93FGPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50135286(CHEMBL3745885)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human TTBK2 using MBP substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24Q7WT8PubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602927(CHEMBL5193908)copy SMILES
Affinity DataIC50: 1.19E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602902(CHEMBL5208571)copy SMILES
Affinity DataIC50: 1.37E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602894(CHEMBL5186604)copy SMILES
Affinity DataIC50: 1.39E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
TargetTau-tubulin kinase 2(Homo sapiens (Human))TBA
LigandPNGBDBM50602890(CHEMBL5198629)copy SMILES
Affinity DataIC50: 1.57E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2R215GVPubMed
Displayed 1 to 50 (of 56 total ) | Next | Last >>
Jump to: