Compile Data Set for Download or QSAR
Found 325 Enz. Inhib. hit(s) with Target = 'Protein-lysine 6-oxidase'
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM50526737(CHEMBL4528500 | US10807974, Example 82 | US1099508...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:Cell Culture and TransfectionAll cell lines used in this study was purchased from American Type Culture Collection (ATCC). Mycoplasma contamination w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Mus musculus)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM50526737(CHEMBL4528500 | US10807974, Example 82 | US1099508...)copy SMILEScopy InChI
Affinity DataIC50: 180nMAssay Description:To produce MDCK cysts, cells were cultured on Matrigel (Corning) with 2% Matrigel supplemented in DMEM with 10% FBS. Cysts were allowed to form for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM50526721(CHEMBL4444163 | US10807974, Example 111 | US109950...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Cell Culture and TransfectionAll cell lines used in this study was purchased from American Type Culture Collection (ATCC). Mycoplasma contamination w...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Mus musculus)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM50526721(CHEMBL4444163 | US10807974, Example 111 | US109950...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:To produce MDCK cysts, cells were cultured on Matrigel (Corning) with 2% Matrigel supplemented in DMEM with 10% FBS. Cysts were allowed to form for 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469007(US10807974, Example 16 | US10995088, Example 16 | ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469007(US10807974, Example 16 | US10995088, Example 16 | ...)copy SMILEScopy InChI
Affinity DataIC50: 300nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633180(4-((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-2-methyl...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633181(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(N,N-di...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633197(N,N′-((((((((((5-(1-((Z)-4-amino-2-fluorobut...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633202(N,N′-((((5-(1-((Z)-4-amino-2-fluorobut-2-en-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633203(5-(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(N,N...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633204(5-(4-(1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-3-(3-(...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633224(4-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633227(2-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633233(3-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633244(3-(((Z)-4-amino-2-fluorobut-2-en-1-yl)sulfonyl)-N-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633245((3aS,4S,6aR)-4-(5-(4-(3-(3-(((Z)-4-amino-2-fluorob...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633246((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((5...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633247((3aS,3a'S,4S,4'S,6aR,6a′R)-4,4′-(((((3...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633248((3aS,4S,6aR)-4-(4-(4-(3-((3-(((Z)-4-amino-2-fluoro...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633249(N-((1-(4-(((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM633250(N-((1-(4-(((1-((Z)-4-amino-2-fluorobut-2-en-1-yl)-...)copy SMILES
Affinity DataIC50: 300nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM50058655(1,1',1'',1'''-[disulfanediylbis(carbonothioylnitri...)copy SMILEScopy InChI
Affinity DataIC50: 320nMAssay Description:Inhibition of recombinant human LOX expressed in HEK293 cells using diaminopentane as substrate preincubated for 30 mins followed by substrate additi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28P6366PubMed
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469005(US10807974, Example 9 | US10995088, Example 9 | US...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469005(US10807974, Example 9 | US10995088, Example 9 | US...)copy SMILEScopy InChI
Affinity DataIC50: 340nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM50505633(CHEMBL4448713)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4GJ2PubMed
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM50505649(CHEMBL4439437)copy SMILEScopy InChI
Affinity DataIC50: 398nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4GJ2PubMed
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469011(US10807974, Example 27 | US10995088, Example 27 | ...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469011(US10807974, Example 27 | US10995088, Example 27 | ...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469032(US10807974, Example 43 | US10995088, Example 43 | ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469032(US10807974, Example 43 | US10995088, Example 43 | ...)copy SMILEScopy InChI
Affinity DataIC50: 420nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469023(US10807974, Example 39 | US10995088, Example 39 | ...)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469023(US10807974, Example 39 | US10995088, Example 39 | ...)copy SMILEScopy InChI
Affinity DataIC50: 440nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469008(US10807974, Example 17 | US10995088, Example 17 | ...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469019(US10807974, Example 35 | US10995088, Example 35 | ...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469008(US10807974, Example 17 | US10995088, Example 17 | ...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469019(US10807974, Example 35 | US10995088, Example 35 | ...)copy SMILEScopy InChI
Affinity DataIC50: 450nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469024(US10807974, Example 40 | US10995088, Example 40 | ...)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469024(US10807974, Example 40 | US10995088, Example 40 | ...)copy SMILEScopy InChI
Affinity DataIC50: 470nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469004(US10807974, Example 5 | US10995088, Example 5 | US...)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469004(US10807974, Example 5 | US10995088, Example 5 | US...)copy SMILEScopy InChI
Affinity DataIC50: 480nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM50505657(CHEMBL4467234)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4GJ2PubMed
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM50505659(CHEMBL4459524)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4GJ2PubMed
TargetProtein-lysine 6-oxidase(Bos taurus)TBA
LigandPNGBDBM50505655(CHEMBL4441299)copy SMILEScopy InChI
Affinity DataIC50: 501nMAssay Description:Inhibition of LOX in bovine aorta using putrescine as substrate preincubated with enzyme for 30 mins followed by substrate addition and measured ever...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4GJ2PubMed
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469027(US10807974, Example 12 | US10995088, Example 12 | ...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469027(US10807974, Example 12 | US10995088, Example 12 | ...)copy SMILEScopy InChI
Affinity DataIC50: 510nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Sus scrofa)
The Institute of Cancer Research: Royal Cancer Hospital

US Patent
LigandPNGBDBM469018(US10807974, Example 34 | US10995088, Example 34 | ...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:LOX enzyme was obtained from pig skin by the method of Shackleton et al 1990.More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2TH8QS8US Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469018(US10807974, Example 34 | US10995088, Example 34 | ...)copy SMILEScopy InChI
Affinity DataIC50: 530nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM50232678(CHEBI:27413 | CHEMBL1618272 | US10717734, Compound...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:Inhibition of full length recombinant human LOX expressed in HEK cells assessed as reduction in H2O2 production using DAP as substrate preincubated f...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542QV6PubMed
TargetProtein-lysine 6-oxidase(Homo sapiens (Human))
THE INSTITUTE OF CANCER RESEARCH: ROYAL CANCER HOSPITAL

US Patent
LigandPNGBDBM469010(US10807974, Example 26 | US10995088, Example 26 | ...)copy SMILEScopy InChI
Affinity DataIC50: 550nMAssay Description:The following reagents were prepared:Reagents500 mM CHES, pH 9 (with NaOH), filtered (MW=207.29)20.7 g in 200 ml in dH2O10% Pluronic F-127 (store at ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2125WSKUS Patent
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