Affinity DataIC50: 0.0200nMAssay Description:Antibacterial activity against Streptococcus faecalis assessed as growth inhibitionMore data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 5nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
Ligand Info
In DepthDetails
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 17nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 24nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 28.6nMAssay Description:Antibacterial activity against Streptococcus faecalis by broth microdilution techniqueMore data for this Ligand-Target Pair
Affinity DataIC50: 36.2nMAssay Description:Antibacterial activity against Enterococcus faecalis MTCC 439 incubated overnight by broth dilution techniqueMore data for this Ligand-Target Pair
Affinity DataIC50: 41.4nMAssay Description:Antibacterial activity against gram positive bacteria Enterococcus faecalis was determined by twofold Micro-broth dilution assayMore data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 49nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 51nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 58nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 73nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 130nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 130nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 167nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 200nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 219nMAssay Description:Concentration (IC50) to inhibit the growth of Streptococcus faecalis.More data for this Ligand-Target Pair
Affinity DataIC50: 401nMAssay Description:Concentration (IC50) to inhibit the growth of Streptococcus faecalis.More data for this Ligand-Target Pair
Affinity DataIC50: 445nMAssay Description:Antibacterial activity against Streptococcus faecalis by broth microdilution techniqueMore data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 450nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 603nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-sensitive Enterococcus faecalis ATCC 29212 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of P450 sccMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis AUS-RBWH-VRE-01 assessed as reduction in fungal growth incubated for 24 hrs...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Antibacterial activity against vancomycin-sensitive Enterococcus faecalis 12-5 after 18 hrs by broth microdilution methodMore data for this Ligand-Target Pair
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of cholesterol side chain cleavage cytochrome P450More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 1.30E+3nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 1.40E+3nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.57E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth dilution assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.60E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis AUS-RBWH-VRE-01 assessed as reduction in fungal growth incubated for 24 hrs...More data for this Ligand-Target Pair
TargetCholesterol side-chain cleavage enzyme, mitochondrial(Bos taurus (Bovine))
CORTENDO AB (PUBL)
US Patent
CORTENDO AB (PUBL)
US Patent
Affinity DataIC50: 1.80E+3nMAssay Description:Cyp11 assay protocol: AD293 cells that stably over-express recombinant CYP-11 were seeded in 96 well plates coated with poly D-lysine (15,000 cell pe...More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Antibacterial activity against vancomycin-resistant Enterococcus faecalis ATCC 51299 after 18 hrs by broth dilution assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.17E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.23E+3nMAssay Description:Antibacterial activity against gram positive bacteria Enterococcus faecalis was determined by twofold Micro-broth dilution assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+3nMAssay Description:Antibacterial activity against low level vancomycin-resistant Enterococcus faecalis ATCC 51299 by plate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.29E+3nMAssay Description:Antimicrobial activity against Enterococcus faecalis assessed as inhibition of biofilm formation after 20 hrs by crystal violet staining analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+3nMAssay Description:Antibacterial activity against Enterococcus faecalis ATCC 51299 assessed as growth inhibition using fresh sample in DMSO by CLSI methodMore data for this Ligand-Target Pair