Compile Data Set for Download or QSAR
Found 18 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-4'
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185644((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)copy SMILEScopy InChI
Affinity DataKi:  6.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185624((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)copy SMILEScopy InChI
Affinity DataKi:  7.80E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185630(CHEMBL210871 | Pam-YDL)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185625(CHEMBL380390 | pAM-FKF)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185628((S)-2-{(S)-4-carboxy-2-[(S)-2-dodecanoylamino-3-(4...)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185618((S)-4-((S)-1-carboxy-2-(4-hydroxyphenyl)ethylamino...)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185645((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-3-hydroxy-2-(...)copy SMILEScopy InChI
Affinity DataKi:  8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185646(CHEMBL207452 | Pam-YKF)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185643((S)-2-{(S)-4-carboxy-2-[(S)-2-hexadecanoylamino-3-...)copy SMILEScopy InChI
Affinity DataKi: >8.00E+4nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Saccharomyces cerevisiae)
CNRS-Université Paris VI

Curated by ChEMBL
LigandPNGBDBM50185633((S)-2-((S)-6-amino-2-((S)-2-((2S,3R)-2-((S)-2-((2S...)copy SMILEScopy InChI
Affinity DataKi:  3.15E+5nMAssay Description:Inhibition of trypsin like activity of yeast 20S proteasomeMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q280527ZPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50577134(CHEMBL4877708)copy SMILES
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WZNPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50577131(CHEMBL4855915)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WZNPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50007203(CHEMBL3237875)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WZNPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50577116(CHEMBL4872258)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WZNPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50577133(CHEMBL4870115)copy SMILES
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human trypsin-like activity of 20s proteasome beta 2c subunit using SUC-KQL-AMC as flurogenic substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BR8WZNPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50604328(CHEMBL5180795)copy SMILES
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1077ZPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50604305(CHEMBL5209480)copy SMILES
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1077ZPubMed
TargetProteasome subunit beta type-4(Homo sapiens (Human))TBA
LigandPNGBDBM50604324(CHEMBL5183361)copy SMILES
Affinity DataIC50: 4.00E+4nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2J1077ZPubMed