Compile Data Set for Download or QSAR
Found 46 of ic50 for UniProtKB: P00772
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50312532(CHEMBL1077010 | molassamide)copy SMILEScopy InChI
Affinity DataIC50: 32nMAssay Description:Inhibition of pig pancreatic elastase preincubated for 15 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GH9J4ZPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071973((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071966((R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071968((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 60nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071983((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 190nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50015856(3-Acetoxymethyl-7-formyloxy-5,5,8-trioxo-5lambda*6...)copy SMILEScopy InChI
Affinity DataIC50: 400nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q81C2QPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50015876(7-Acetoxy-3-acetoxymethyl-5,5,8-trioxo-5lambda*6*-...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q81C2QPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071965((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 2.20E+3nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50429202(LYNGBYASTATIN 7)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0J8KPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50479189(CHEBI:66142 | KEMPOPEPTIN A)copy SMILEScopy InChI
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0J8KPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50479190(SOMAMIDE B)copy SMILEScopy InChI
Affinity DataIC50: 4.20E+3nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0J8KPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM50302107(CHEMBL567893 | Grassystatin A)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of porcine pancreatic elastase after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2BG2PXPPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50015857(3-Acetoxymethyl-5,5,8-trioxo-7-phenylacetoxy-5lamb...)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibitory concentration which is required to cause 50% inhibition of Porcine pancreatic elastase (PPE) enzymeMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q81C2QPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237204(Esculin laurate)copy SMILEScopy InChI
Affinity DataIC50: 2.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237205(Esculin myristate)copy SMILEScopy InChI
Affinity DataIC50: 2.50E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237206(Esculin palmitate)copy SMILEScopy InChI
Affinity DataIC50: 3.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-4H-chrome...)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237207(Esculin stearate)copy SMILEScopy InChI
Affinity DataIC50: 6.00E+4nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50479191(KEMPOPEPTIN B)copy SMILEScopy InChI
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibition of pig pancreatic elastaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29W0J8KPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237184(Rutin)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237198(Phloridzin)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237203(Esculin)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071967((R)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 2.06E+5nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237208(4-Guanidinobenzoate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237196(Rutin arachidonate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237195(Rutin linolenate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237194(Rutin linoleate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237197(Rutin erucate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237199(Phloridzin laurate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237200(Phloridzin myristate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237202(Phloridzin stearate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237201(Phloridzin palmitate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237185(Rutin butyrate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237186(Rutin caproate | Rutin capronate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237187(Rutin caprylate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237186(Rutin caproate | Rutin capronate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237193(Rutin oleate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237192(Rutin stearate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237191(Rutin palmitate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237190(Rutin myristate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1(Sus scrofa (Pig))
Smithsonian Marine Station at Ft. Pierce

Curated by ChEMBL
LigandPNGBDBM237189(Rutin laurate)copy SMILEScopy InChI
Affinity DataIC50: 5.00E+5nMpH: 8.0Assay Description:The rate of hydrolysis of the substrates (0.3 mM) by trypsin (18 U/ml), thrombin (12.5 NIH U/ml), urokinase (62500 IU/ml) and elastase (8.4 U/ml) was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RR1X5TPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50284214(Acetic acid 2,4-dioxo-9-phenethyl-1,2,4,9-tetrahyd...)copy SMILEScopy InChI
Affinity DataIC50: 8.33E+5nMAssay Description:Inhibitory activity against porcine pancreatic elastase using Suc-Ala-Ala-Ala-pNA (416 uM) as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6C4C
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50284202(Acetic acid 2,4-dioxo-9-(3-phenyl-propyl)-1,2,4,9-...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against porcine pancreatic elastase using Suc-Ala-Ala-Ala-pNA (416 uM) as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6C4C
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071975((S)-3-((S)-2-Acetylamino-3-carboxy-propionylamino)...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50284206(Acetic acid 9-butyl-2,4-dioxo-1,2,4,9-tetrahydro-[...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against porcine pancreatic elastase using Suc-Ala-Ala-Ala-pNA (416 uM) as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27W6C4C
TargetChymotrypsin-like elastase family member 1/2A(Sus scrofa (Pig))
Boehringer Ingelheim (Canada) Ltd

Curated by ChEMBL
LigandPNGBDBM50071970((R)-2-{[1-((S)-2-{(2S,3S)-2-[(R)-2-((S)-2-Acetylam...)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+6nMAssay Description:Compound was tested for inhibition of porcine pancreatic elastase (PPE)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2V69HRXPubMed