Compile Data Set for Download or QSAR
Found 93 of ki for UniProtKB: P05129
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391386(CHEMBL2148106)copy SMILEScopy InChI
Affinity DataKi:  0.380nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q200036JPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327943(Aplysiatoxin | CHEMBL1256416)copy SMILEScopy InChI
Affinity DataKi:  0.630nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2H04PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50587724(CHEMBL5175742)copy SMILES
Affinity DataKi:  0.650nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q2260PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50493217(DEMETHOXYDEBROMOAPLYSIATOXIN)copy SMILEScopy InChI
Affinity DataKi:  0.690nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domain (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VD72CXPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057514((10S,13S)-13-Hydroxymethyl-10-isopropyl-9-methyl-5...)copy SMILEScopy InChI
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319TZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50133236(CHEMBL337834 | Tetradecanedioic acid ((S)-5-hydrox...)copy SMILEScopy InChI
Affinity DataKi:  1.5nMAssay Description:Inhibition of human Protein kinase C gamma with [Ca2+]More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2GF0SX2PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)copy SMILEScopy InChI
Affinity DataKi:  1.60nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VM4BHZPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50097750(Butyric acid (1aR,1bS,4aS,7aR,7bR,8R,9R,9aS)-9-but...)copy SMILEScopy InChI
Affinity DataKi:  1.80nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VM4BHZPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057512((1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-4a,7b-dihydroxy-3-...)copy SMILEScopy InChI
Affinity DataKi:  2.90nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VM4BHZPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)copy SMILEScopy InChI
Affinity DataKi:  4.90nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D799PVPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50097750(Butyric acid (1aR,1bS,4aS,7aR,7bR,8R,9R,9aS)-9-but...)copy SMILEScopy InChI
Affinity DataKi:  5.20nMAssay Description:Displacement of 3[H]PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2VM4BHZPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391388(CHEMBL2148108)copy SMILEScopy InChI
Affinity DataKi:  5.5nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q200036JPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50391387(CHEMBL2148107)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q200036JPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  12nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249959(CHEMBL522428 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  16nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  19.4nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319TZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50368315(PROSTRATIN)copy SMILEScopy InChI
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26Q2260PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249958(CHEMBL489520 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  32nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  35nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445M7QPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]PDBu binding to PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q200036JPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327946(1S,3R,5R,9R,13R)-9-Hydroxymethyl-3-[4-(3-hydroxy-p...)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2H04PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50229772(1-hexylindolactam-V | CHEMBL399981)copy SMILEScopy InChI
Affinity DataKi:  39nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445M7QPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)copy SMILEScopy InChI
Affinity DataKi:  40.7nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319TZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)copy SMILEScopy InChI
Affinity DataKi:  43nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D799PVPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  51nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445M7QPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  59nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2445M7QPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374190(CHEMBL271403)copy SMILEScopy InChI
Affinity DataKi:  61nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5W85PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249885(CHEMBL492118 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  78nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50327944((1S,3R,5R,9R,13R)-9-Hydroxymethyl-16,16-dimethyl-3...)copy SMILEScopy InChI
Affinity DataKi:  80nMAssay Description:Inhibition of [3H]PDBu binding to PKC gamma C1A peptideMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2FJ2H04PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  138nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7NZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  138nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C eta C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QV3KRSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5W85PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50249884(CHEMBL523155 | [2-(Hydroxymethyl)-4-(methylethylid...)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Displacement of [3H]PDBu form human PKCgamma in presence of plasma membrane lipid mimetic mixtureMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2862GB6PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC gamma expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2319TZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057510((2S,5S)-8-Decyl-5-hydroxymethyl-2-isopropyl-1-meth...)copy SMILEScopy InChI
Affinity DataKi:  151nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QV3KRSPubMed
LigandPNGBDBM50368315(PROSTRATIN)copy SMILEScopy InChI
Affinity DataKi:  190nMAssay Description:Displacement of [3H]PDBu binding to Protein kinase C of CEM cells with 10% fetal calf serumMore data for this Ligand-Target Pair
LigandPNGBDBM50281846((2R,3R)-2-Hydroxymethyl-5-oxo-4-tridec-(E)-ylidene...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of [20-3H]phorbol-12,13-dibutyrate (PDBU) binding to protein kinase CMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20C4VQP
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099064(CHEMBL368720 | Dodecanoic acid (3S,3aR,8R,8aS)-3-h...)copy SMILEScopy InChI
Affinity DataKi:  209nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D799PVPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5W85PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50463479(CHEMBL4249925)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of PKCgamma (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2ZC85HXPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  213nMAssay Description:Displacement of [3H]- PDBu from Protein kinase C gamma C1b domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7NZSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50057511((+/-)-indolactum-V 13-Hydroxymethyl-10-isopropyl-9...)copy SMILEScopy InChI
Affinity DataKi:  213nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to Protein kinase C gamma C1a domainMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2QV3KRSPubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374190(CHEMBL271403)copy SMILEScopy InChI
Affinity DataKi:  225nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1B domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5W85PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50374191(CHEMBL261387)copy SMILEScopy InChI
Affinity DataKi:  234nMAssay Description:Displacement of [3H]PDBu from PKCgamma C1A domainMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2XS5W85PubMed
TargetProtein kinase C gamma type(Homo sapiens (Human))
Kyoto University

Curated by ChEMBL
LigandPNGBDBM50099065((3S,3aR,8R,8aS)-6-Dec-1-ynyl-3-hydroxymethyl-8-iso...)copy SMILEScopy InChI
Affinity DataKi:  279nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C gammaMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2D799PVPubMed
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