Compile Data Set for Download or QSAR
Found 14 of ec50 for UniProtKB: P17252
LigandPNGBDBM50519087(CHEMBL3741746)copy SMILEScopy InChI
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959MZJPubMed
LigandPNGBDBM50519063(CHEMBL4587471)copy SMILEScopy InChI
Affinity DataEC50:  0.550nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959MZJPubMed
LigandPNGBDBM50519068(CHEMBL4575056)copy SMILEScopy InChI
Affinity DataEC50:  0.600nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959MZJPubMed
LigandPNGBDBM50519085(CHEMBL4444766)copy SMILEScopy InChI
Affinity DataEC50: >3.90nMAssay Description:Agonist activity at Protein kinase C in human U1 cells infected with HIV-1 NL4-3 assessed as induction of HIV-1 p24 production after 72 hrs by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2959MZJPubMed
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)copy SMILEScopy InChI
Affinity DataEC50:  9.5nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6N3MPubMed
LigandPNGBDBM50470108(AGN 204332 | Ingenol Mebutate | PEP-005 | PEP005 |...)copy SMILEScopy InChI
Affinity DataEC50:  73nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
LigandPNGBDBM50368315(PROSTRATIN)copy SMILEScopy InChI
Affinity DataEC50:  910nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
LigandPNGBDBM50470110(CHEMBL4071723)copy SMILEScopy InChI
Affinity DataEC50:  5.04E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6N3MPubMed
LigandPNGBDBM50470109(CHEMBL4104319)copy SMILEScopy InChI
Affinity DataEC50:  6.08E+3nMAssay Description:Activation of PKC in human platelet assessed as induction of platelet aggregation measured within 15 mins by tribidimetric methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24T6N3MPubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Houston

Curated by ChEMBL
LigandPNGBDBM23928(1,3-dimethoxy-5-[(E)-2-(4-methoxyphenyl)ethenyl]be...)copy SMILEScopy InChI
Affinity DataEC50:  1.56E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GN9PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Houston

Curated by ChEMBL
LigandPNGBDBM50099066(CHEMBL279115 | phorbol 13-acetate 12-myristate)copy SMILEScopy InChI
Affinity DataEC50:  1.70E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GN9PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Houston

Curated by ChEMBL
LigandPNGBDBM50351474(CHEMBL1819531)copy SMILEScopy InChI
Affinity DataEC50:  2.98E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GN9PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Houston

Curated by ChEMBL
LigandPNGBDBM50351475(CHEMBL1819528)copy SMILEScopy InChI
Affinity DataEC50:  5.04E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GN9PubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
University of Houston

Curated by ChEMBL
LigandPNGBDBM23926((E)-resveratrol | 5-[(E)-2-(4-hydroxyphenyl)etheny...)copy SMILEScopy InChI
Affinity DataEC50:  5.78E+6nMAssay Description:Binding affinity to recombinant C1 domain of PKCalpha expressed in Escherichia coli BL21 (DE3) after 45 mins by fluorescence quenching assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7GN9PubMed