Compile Data Set for Download or QSAR
Found 1027 of ic50 for UniProtKB: P26618
LigandPNGBDBM50408387(CHEMBL5268482)copy SMILEScopy InChI
Affinity DataIC50: 0.0400nMAssay Description:Antagonist activity at human P2X7 receptor transfected in THP1 cells assessed as inhibition of benzoyl-ATP-induced changes in plasma membrane pore fo...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50477652(CHEMBL250790)copy SMILEScopy InChI
Affinity DataIC50: 0.0900nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608338(CHEMBL5268427)copy SMILES
Affinity DataIC50: 0.140nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50518950(CHEMBL4468881)copy SMILEScopy InChI
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608648(CHEMBL5286715)copy SMILES
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608647(CHEMBL5267724)copy SMILES
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608649(CHEMBL5290499)copy SMILES
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608650(CHEMBL5271348)copy SMILES
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608646(CHEMBL5288936)copy SMILES
Affinity DataIC50: 0.210nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50450068(CHEMBL5275288)copy SMILEScopy InChI
Affinity DataIC50: 0.216nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50450067(CHEMBL5279750)copy SMILEScopy InChI
Affinity DataIC50: 0.216nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408386(CHEMBL5287343)copy SMILEScopy InChI
Affinity DataIC50: 0.260nMAssay Description:Antagonist activity at human P2X7 receptor transfected in THP1 cells assessed as inhibition of benzoyl-ATP-induced changes in plasma membrane pore fo...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50411638(CHEMBL404371)copy SMILEScopy InChI
Affinity DataIC50: 0.5nMAssay Description:Antagonist activity at human P2X7 receptor transfected in THP1 cells assessed as inhibition of benzoyl-ATP-induced changes in plasma membrane pore fo...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50226181((3R,4S,5R,6R)-5-hydroxy-6-(4-hydroxy-3-(4-hydroxy-...)copy SMILEScopy InChI
Affinity DataIC50: 0.650nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50407412(CHEMBL5269793)copy SMILEScopy InChI
Affinity DataIC50: 0.700nMAssay Description:Activity at Histamine H2 receptor using functional H2 receptor assay on guinea pig atriumMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 0.770nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50000334(6,7-Dichloro-1,5-dihydro-imidazo[2,1-b]quinazolin-...)copy SMILEScopy InChI
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50608668(CHEMBL5282942)copy SMILES
Affinity DataIC50: 0.950nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50613596(CHEMBL5272356)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
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LigandPNGBDBM50193093(RGB-286638)copy SMILEScopy InChI
Affinity DataIC50: 1nMAssay Description:Ability to displace [3H]glycine from strychnine-insensitive glycine receptorMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50613594(CHEMBL5275755)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50613593(CHEMBL5285324)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50613595(CHEMBL5272100)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50613597(CHEMBL5270626)copy SMILES
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50613099(CHEMBL5288212)copy SMILES
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50239948(CHEMBL4071326 | US9850225, Example 1166)copy SMILEScopy InChI
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50610586(CHEMBL5280445)copy SMILES
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50450065(CHEMBL5286795)copy SMILEScopy InChI
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50614520(CHEMBL5271228)copy SMILES
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608645(CHEMBL4535844)copy SMILES
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50608666(CHEMBL5267457)copy SMILES
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50450066(CHEMBL5283958)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50408479(CHEMBL5180503)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMAssay Description:Antagonist activity at human P2X7 receptor transfected in THP1 cells assessed as inhibition of benzoyl-ATP-induced changes in plasma membrane pore fo...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM21691(1-ethyl-7-methyl-4-oxo-1,4-dihydro-1,8-naphthyridi...)copy SMILEScopy InChI
Affinity DataIC50: 1.70nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50410546(CHEMBL26159)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Inhibitory activity against Dihydrofolate reductase in Neisseria gonorrhoeaeMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50448498(BMS-791325 | Beclabuvir)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMMore data for this Ligand-Target Pair
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LigandPNGBDBM50241662(CHEMBL4104741)copy SMILEScopy InChI
Affinity DataIC50: 1.80nMAssay Description:Dissociation constant against VEGF (vascular endothelial growth factor) was determined.More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50193093(RGB-286638)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Blocking activity against Beta-1 adrenergic receptor in spontaneously beating guinea pig atrial preparationsMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50512074(CHEMBL4575813)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Antagonist activity at M3 receptor in Dunkin-Hartley guinea pig trachea assessed as inhibition of methacholine-induced airway smooth muscle contracti...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM50322535(3-(imidazo[1,2-b]pyridazin-3-ylethynyl)-4-methyl-N...)copy SMILEScopy InChI
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 2nMAssay Description:Inhibition of Platelet-derived growth factor receptor in P19 cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2765DVXPubMed
LigandPNGBDBM50239946(CHEMBL4084368)copy SMILEScopy InChI
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50608667(CHEMBL5271201)copy SMILES
Affinity DataIC50: 2.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)copy SMILEScopy InChI
Affinity DataIC50: 2.40nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50404385(CHEMBL5273069)copy SMILEScopy InChI
Affinity DataIC50: 2.5nMAssay Description:In vitro antagonism of the 5-HT-3 receptor determined by inhibition of 5-HT-induced depolarization of the isolated rat vagus nerve.More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM8131(N-(4-Isopropylphenyl)-4-pyrazolo[1,5-b]pyridazin-3...)copy SMILEScopy InChI
Affinity DataIC50: 2.70nMAssay Description:The compound was evaluated for its relative binding affinity against mutant N131A scytalone dehydratase; Relative KiMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM21690(1-cyclopropyl-6-fluoro-4-oxo-7-(piperazin-1-yl)-1,...)copy SMILEScopy InChI
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50239948(CHEMBL4071326 | US9850225, Example 1166)copy SMILEScopy InChI
In DepthDetails
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