Compile Data Set for Download or QSAR
Found 8 of ic50 for UniProtKB: P28472
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50106149(1-(2,6-Dichloro-4-trifluoromethyl-phenyl)-4-(3-tri...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]-EBOB binding to human GABA-A receptor beta3 subunit (range 1-28)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KS6QTJPubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50106148(5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]-EBOB binding to drosophila GABA-A receptor (range 1-28)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KS6QTJPubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50106148(5-amino-1-[2,6-dichloro-4-(trifluoromethyl)phenyl]...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]-EBOB binding to drosophila GABA-A receptor (range 1-28)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KS6QTJPubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50106149(1-(2,6-Dichloro-4-trifluoromethyl-phenyl)-4-(3-tri...)copy SMILEScopy InChI
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]-EBOB binding to human GABA-A receptor beta3 subunit (range 1-28)More data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2KS6QTJPubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50395121(CHEMBL2163548)copy SMILEScopy InChI
Affinity DataIC50: 3.90E+3nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B03MXPubMed
LigandPNGBDBM50580362(CHEMBL5086854)copy SMILES
Affinity DataIC50: 5.50E+3nMAssay Description:Negative allosteric modulation activity at human GABAA alpha3beta3gamma2 stably expressed in HEK cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2TX3K7PPubMed
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50055935(5-Ethyl-5-(1-methylbutyl)-2,4,6(1H,3H,5H)-pyrimidi...)copy SMILEScopy InChI
Affinity DataIC50: 8.80E+4nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B03MXPubMedDrugBank
TargetGamma-aminobutyric acid receptor subunit beta-3(Homo sapiens (Human))
University of California

Curated by ChEMBL
LigandPNGBDBM50395120(CHEMBL2163549)copy SMILEScopy InChI
Affinity DataIC50: 1.70E+5nMAssay Description:Displacement of [3H]R-(-)-14 from human FLAG-tagged beta3 GABA A receptor expressed in HEK293S cellsMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25B03MXPubMed