Compile Data Set for Download or QSAR
Found 8 of ki for UniProtKB: P29703
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298243((2E,6E)-8-(2-diazo-3,3,3-trifluoropropanoyloxy)-3,...)copy SMILEScopy InChI
Affinity DataKi:  200nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2PCHPubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289981(Prenyl pyrophosphate analogue | {[(2E,6E)-8-[(3-be...)copy SMILEScopy InChI
Affinity DataKi:  380nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P3X
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298245(4-Benzoylbenzylphosphonic((2E,6E)-3,7,11-trimethyl...)copy SMILEScopy InChI
Affinity DataKi:  480nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2PCHPubMed
TargetProtein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae)
University of Minnesota

Curated by ChEMBL
LigandPNGBDBM50298242((E)-4-(3-benzoylbenzyloxy)-3-methylbut-2-enyl diph...)copy SMILEScopy InChI
Affinity DataKi:  610nMAssay Description:Inhibition of Saccharomyces cerevisiae protein farnesyltransferase assessed as farnsylation of N-dansyl-GCVIAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2PCHPubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289982(Prenyl pyrophosphate analogue)copy SMILEScopy InChI
Affinity DataKi:  700nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P3X
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289979(Prenyl pyrophosphate analogue | {[(2E)-4-[(3-benzo...)copy SMILEScopy InChI
Affinity DataKi:  960nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P3X
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50289978(Prenyl pyrophosphate analogue | {[(2E)-4-[(3-benzo...)copy SMILEScopy InChI
Affinity DataKi:  6.00E+3nMAssay Description:Inhibition of yeast Farnesyl transferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2542P3X
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Saccharomyces cerevisiae (Baker's yeast))
TBA

Curated by ChEMBL
LigandPNGBDBM50144314((2E,4E,6E,8E)-3,7,11-trimethyldodeca-2,4,6,8,10-pe...)copy SMILEScopy InChI
Affinity DataKi:  8.80E+3nMAssay Description:Dissociation constant against yeast farnesyltransferaseMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S181Z3PubMed