Compile Data Set for Download or QSAR
Found 200 of ec50 for UniProtKB: P48039
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM103443(US8552037, 90)copy SMILEScopy InChI
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human MT1 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7M2BPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50347588(CHEMBL1802025)copy SMILEScopy InChI
Affinity DataEC50:  0.0210nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2PN3PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.0220nMAssay Description:Agonist activity at human MT1 expressed in CHO-K1 cells assessed as inhibition of forskolin-induced cAMP accumulation incubated for 30 mins by AlphaS...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q25H7M2BPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.0260nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as decrease in forskolin-stimulated cAMP release after 30 mins by multilabel p...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2HT2PN3PubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463444(US10781182, Compound IA2-121 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0350nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463443(US10781182, Compound IA2-120 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0360nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575514(CHEMBL4852440)copy SMILES
Affinity DataEC50:  0.0370nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575511(CHEMBL4859677)copy SMILES
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575513(CHEMBL4873903)copy SMILES
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575512(CHEMBL4854625)copy SMILES
Affinity DataEC50:  0.0420nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50464413(CHEMBL4281712)copy SMILEScopy InChI
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463447(US10781182, Compound IA2-143 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.0630nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.0692nMMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.0980nMAssay Description:Agonist activity at human melatonin receptor-1 transfected in CHO cell membranes after 1 hr by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2JM2CDGPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463444(US10781182, Compound IA2-121 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575516(CHEMBL4874954)copy SMILES
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50114703(CHEMBL287560 | N-[2-(5-Methoxy-2-phenyl-benzofuran...)copy SMILEScopy InChI
Affinity DataEC50:  0.170nMAssay Description:Intrinsic activity evaluated on [35S]-GTP -gamma-S binding in Chinese hamster ovarian (CHO) cells, stably expressing human Melatonin receptor type 1AMore data for this Ligand-Target Pair
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2Q52P0WPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463443(US10781182, Compound IA2-120 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.180nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50464412(CHEMBL4278248)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575512(CHEMBL4854625)copy SMILES
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50464409(CHEMBL4283539)copy SMILEScopy InChI
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463445(US10781182, Compound IA2-140 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.233nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575510(CHEMBL4867553)copy SMILES
Affinity DataEC50:  0.240nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463447(US10781182, Compound IA2-143 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50598933(CHEMBL5174929)copy SMILES
Affinity DataEC50:  0.257nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMed
TargetMelatonin receptor type 1A/1B(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50149182(CHEMBL124577 | N-[3-(2-Methyl-benzooxazol-7-yl)-pr...)copy SMILEScopy InChI
Affinity DataEC50:  0.260nMAssay Description:Agonist activity for its ability to inhibit forskolin-stimulated cAMP accumulation against MT1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2S75FSRPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575514(CHEMBL4852440)copy SMILES
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575511(CHEMBL4859677)copy SMILES
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575513(CHEMBL4873903)copy SMILES
Affinity DataEC50:  0.420nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50598931(CHEMBL5209359)copy SMILES
Affinity DataEC50:  0.447nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50598931(CHEMBL5209359)copy SMILES
Affinity DataEC50:  0.589nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50153420(1N-[2-[2-(4-phenylbutyl)benzo[b]furan-4-yl]-(1R,2R...)copy SMILEScopy InChI
Affinity DataEC50:  0.600nMAssay Description:Agonist activity towards human Melatonin receptor type 1A was determined by its ability to inhibit forskolin stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2M044XGPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50598930(CHEMBL5173623)copy SMILES
Affinity DataEC50:  0.617nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575517(CHEMBL4869463)copy SMILES
Affinity DataEC50:  0.75nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50230955(CHEMBL4102177)copy SMILEScopy InChI
Affinity DataEC50:  0.800nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24F1SZSPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50117899(CHEMBL3612604)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Intrinsic activity at human MT1 receptor transfected in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q20R9R6DPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50464400(CHEMBL4293386)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50464399(CHEMBL4278446)copy SMILEScopy InChI
Affinity DataEC50:  0.900nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CC13BXPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM463446(US10781182, Compound IA2-142 | US11091445, Compoun...)copy SMILEScopy InChI
Affinity DataEC50:  0.937nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in forskolin induced cAMP production incubated at 37 degreeC by Hi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50575515(CHEMBL4872217)copy SMILES
Affinity DataEC50:  0.970nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells assessed as increase in cAMP levels incubated at 28 degreeC by cellular dielectric spec...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z03CZJPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Agonist activity at MT1 receptor (unknown origin) expressed in HEK293 cells by Fluo-8 dye-based calcium assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q290276RPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50144226(CHEMBL3758679)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50144224(CHEMBL3759816)copy SMILEScopy InChI
Affinity DataEC50:  1nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2VM4F3TPubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50598930(CHEMBL5173623)copy SMILES
Affinity DataEC50:  1.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2Z323P9PubMed
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataEC50:  1.40nMAssay Description:Intrinsic activity at human MT1 receptor expressed in CHO cell membranes after 1 hr by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM9019(CHEMBL45 | Melatonin | N-[2-(5-methoxy-1H-indol-3-...)copy SMILEScopy InChI
Affinity DataEC50:  1.5nMAssay Description:Agonist activity at human MT1 receptor expressed in CHO cells by [35S]GTPgamma binding assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27H1JWMPubMedDrugBank
TargetMelatonin receptor type 1A(Homo sapiens (Human))TBA
LigandPNGBDBM50035179(Agomelatine | CHEMBL10878 | N-[2-(7-Methoxy-naphth...)copy SMILEScopy InChI
Affinity DataEC50:  1.56nMAssay Description:Agonist potency determined by [35S]-GTP gamma-S binding assay using CHO cell lines for Melatonin receptor type 1AMore data for this Ligand-Target Pair
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