Compile Data Set for Download or QSAR
Found 158 of ki for UniProtKB: P51946
LigandPNGBDBM498187(US11014911, Example 15 | US11718603, Example 15)copy SMILES
Affinity DataKi:  6.30nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7SJ2
LigandPNGBDBM50528812(CHEMBL4582951)copy SMILEScopy InChI
Affinity DataKi:  17nMAssay Description:Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4T3TPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443446(CHEMBL3087439)copy SMILEScopy InChI
Affinity DataKi:  24nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
LigandPNGBDBM50568690(CHEMBL4870188)copy SMILES
Affinity DataKi:  29nMAssay Description:Inhibition of CDK7/cyclin H/MAT1 (unknown origin) using HYSPTSPSYSPTSPSYSPTSPSKKKK-O substrate incubated for 120 mins measured after 40 mins incubati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z198KPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443449(CHEMBL3087442)copy SMILEScopy InChI
Affinity DataKi:  30nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431337(CHEMBL2348845)copy SMILEScopy InChI
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431340(CHEMBL2348842)copy SMILEScopy InChI
Affinity DataKi:  47nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423756(CHEMBL611995)copy SMILEScopy InChI
Affinity DataKi:  53nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431338(CHEMBL2348844)copy SMILEScopy InChI
Affinity DataKi:  54nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423757(CHEMBL609915)copy SMILEScopy InChI
Affinity DataKi:  60nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
LigandPNGBDBM50528814(CHEMBL4436535)copy SMILEScopy InChI
Affinity DataKi:  63nMAssay Description:Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4T3TPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431339(CHEMBL2348843)copy SMILEScopy InChI
Affinity DataKi:  64nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431355(CHEMBL2348642)copy SMILEScopy InChI
Affinity DataKi:  68nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM8061(2-Anilino-4-(thiazol-5-yl)pyrimidine deriv. 32 | 4...)copy SMILEScopy InChI
Affinity DataKi:  70nM ΔG°:  -9.92kcal/molepH: 7.2 T: 2°CAssay Description:In vitro kinase assay using purified enzyme, was incubated at 30 °C with substrate, and test compounds in the presence of 100 uM ATP/ [gamma-32P...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CJ8BPPPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50229973((4-(2-Amino-4-methylthiazol-5-yl)pyrimidin-2-yl)-(...)copy SMILEScopy InChI
Affinity DataKi:  70nMAssay Description:Inhibition of Cdk7/cyclin HChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2DB82RHPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431353(CHEMBL2348644)copy SMILEScopy InChI
Affinity DataKi:  71nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50570302(CHEMBL4853628)copy SMILES
Affinity DataKi:  89nMAssay Description:Inhibition of recombinant human full length CDK7/Cyclin H using peptide as substrate incubated for 40 mins in presence of [gamma-33P]-ATP by scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2RX9GV5PubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431360(CHEMBL2347597)copy SMILEScopy InChI
Affinity DataKi:  91nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431356(CHEMBL2348641)copy SMILEScopy InChI
Affinity DataKi:  92nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
LigandPNGBDBM50528811(CHEMBL4441405)copy SMILEScopy InChI
Affinity DataKi:  105nMAssay Description:Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4T3TPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443451(CHEMBL3087444)copy SMILEScopy InChI
Affinity DataKi:  110nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431347(CHEMBL2348650)copy SMILEScopy InChI
Affinity DataKi:  111nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50425010(CHEMBL2312183)copy SMILEScopy InChI
Affinity DataKi:  114nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443447(CHEMBL3087440)copy SMILEScopy InChI
Affinity DataKi:  133nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423754(CHEMBL598992)copy SMILEScopy InChI
Affinity DataKi:  140nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
LigandPNGBDBM50568688(CHEMBL4862206)copy SMILES
Affinity DataKi:  142nMAssay Description:Inhibition of CDK7/cyclin H/MAT1 (unknown origin) using HYSPTSPSYSPTSPSYSPTSPSKKKK-O substrate incubated for 120 mins measured after 40 mins incubati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q22Z198KPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50567666(CHEMBL4850615)copy SMILES
Affinity DataKi:  144nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FVFPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM81436(CDK Inhibitor, 9)copy SMILEScopy InChI
Affinity DataKi:  150nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431348(CHEMBL2348649)copy SMILEScopy InChI
Affinity DataKi:  155nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443456(CHEMBL3087432)copy SMILEScopy InChI
Affinity DataKi:  163nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
LigandPNGBDBM498185(US11014911, Example 13 | US11718603, Example 13 | ...)copy SMILES
Affinity DataKi:  177nMMore data for this Ligand-Target Pair
Ligand InfoMCE
PC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q22F7SJ2
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443450(CHEMBL3087443)copy SMILEScopy InChI
Affinity DataKi:  180nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50501587(CHEMBL4066828)copy SMILEScopy InChI
Affinity DataKi:  189nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin) in presence of [gamma-33P]-ATP by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z97XGPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431350(CHEMBL2348647)copy SMILEScopy InChI
Affinity DataKi:  193nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50501588(CHEMBL4102076)copy SMILEScopy InChI
Affinity DataKi:  194nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin) in presence of [gamma-33P]-ATP by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z97XGPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50567665(CHEMBL4855877)copy SMILES
Affinity DataKi:  203nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FVFPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50567652(CHEMBL4878693)copy SMILES
Affinity DataKi:  208nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26W9FVFPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431346(CHEMBL2348651)copy SMILEScopy InChI
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50501598(CHEMBL4103372)copy SMILEScopy InChI
Affinity DataKi:  211nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin) in presence of [gamma-33P]-ATP by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z97XGPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443455(CHEMBL3087448)copy SMILEScopy InChI
Affinity DataKi:  252nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431335(CHEMBL2348847)copy SMILEScopy InChI
Affinity DataKi:  255nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
LigandPNGBDBM50110178(CHEMBL3603847 | US10787436, Compound I-23)copy SMILEScopy InChI
Affinity DataKi:  255nMAssay Description:Competitive irreversible inhibition of CDK7/cyclinH/MAT1 (unknown origin) using 5-FAM YSPTSPSYSPTSPSYSPTSPSKKKK as substrateMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q23F4T3TPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50425011(CHEMBL2312182)copy SMILEScopy InChI
Affinity DataKi:  260nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431336(CHEMBL2348846)copy SMILEScopy InChI
Affinity DataKi:  273nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50501578(CHEMBL4098811)copy SMILEScopy InChI
Affinity DataKi:  282nMAssay Description:Inhibition of CDK7/cyclin H (unknown origin) in presence of [gamma-33P]-ATP by KINOMEscan assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29Z97XGPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431352(CHEMBL2348645)copy SMILEScopy InChI
Affinity DataKi:  286nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50423762(CHEMBL605635)copy SMILEScopy InChI
Affinity DataKi:  300nMAssay Description:inhibition of CDK7/Cyclin H/MAT1More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2377B0RPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431351(CHEMBL2348646)copy SMILEScopy InChI
Affinity DataKi:  302nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50443457(CHEMBL3087433)copy SMILEScopy InChI
Affinity DataKi:  304nMAssay Description:Inhibition of CDK7/Cyclin H (unknown origin) by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q24J0GKSPubMed
TargetCyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University of Nottingham

Curated by ChEMBL
LigandPNGBDBM50431354(CHEMBL2348643)copy SMILEScopy InChI
Affinity DataKi:  316nMAssay Description:Inhibition of human recombinant His6 tagged CDK7/CyclinH/MAT1 expressed in Sf21 insect cells after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q26D5VBBPubMed
Displayed 1 to 50 (of 158 total ) | Next | Last >>
Jump to: