Compile Data Set for Download or QSAR
Found 7 of ic50 for UniProtKB: P52332
TargetTyrosine-protein kinase JAK1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of murine Jak 1 protein kinaseMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM26198(4-tert-butyl-15-fluoro-3,5,10-triazatetracyclo[11....)copy SMILEScopy InChI
Affinity DataIC50: 15nMAssay Description:Inhibition of mouse JAK1Checked by AuthorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50109821(CHEBI:87103 | CHEMBL21156 | US10981896, Compound 4...)copy SMILEScopy InChI
Affinity DataIC50: 15nMMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124147(CHEMBL3622826)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of FLAG-tagged mouse JAK1 expressed in insect Sf9 cells using biotin-EQEDEPEGDYFEWLE-NH2 as substrate by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2K64M0XPubMed
TargetTyrosine-protein kinase JAK1/JAK3(Mus musculus)
Eberhard-Karls-University Tuebingen

Curated by ChEMBL
LigandPNGBDBM153159(BDBM153160 | US8993756, 4-1)copy SMILEScopy InChI
Affinity DataIC50: 70nMAssay Description:Inhibition of JAK3/JAK1 in mouse CTLL-2 cells assessed as reduction in IL2-stimulated STAT5 phosphorylationMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27P91Z2PubMed
TargetNon-receptor tyrosine-protein kinase TYK2/Tyrosine-protein kinase JAK1(Mus musculus)
Janssen Research and Development

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)copy SMILEScopy InChI
Affinity DataIC50: 112nMAssay Description:Inhibition of JAK1/Tyk2-mediated STAT4 phosphorylation in IFNalpha-stimulated mouse whole bloodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK1(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50446982(CHEMBL3116050)copy SMILEScopy InChI
Affinity DataIC50: 260nMAssay Description:Inhibition of Jak1 in mouse BA/F3 cells expressing TEL-Jak1 assessed as inhibition of STAT5 phosphorylation by Western blotting analysisMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2CR5VTMPubMed