Compile Data Set for Download or QSAR
Found 185 of ic50 for UniProtKB: P62813
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482687(CHEMBL426916)copy SMILEScopy InChI
Affinity DataIC50: 7.10nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540736(US11261211, Compound SA-4)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540759(US11261211, Compound SA-39)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540767(US11261211, Compound SA-58)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540748(US11261211, Compound SA-11)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540735(US11261211, Compound SA-2)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540762(US11261211, Compound SA-55)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540766(US11261211, Compound SA-57)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540754(US11261211, Compound SA-15)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540753(US11261211, Compound SA-14)copy SMILES
Affinity DataIC50: 10nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM50000766(CHEMBL12 | DIAZEPAM | US9271961, Diazepam)copy SMILEScopy InChI
Affinity DataIC50: 12nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM23183(5-(aminomethyl)-1,2-oxazol-3-ol | Agarin | CHEMBL2...)copy SMILEScopy InChI
Affinity DataIC50: 16nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q28C9X1XPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM520647(US11147877, Compound 2)copy SMILES
Affinity DataIC50: 20nMAssay Description:Briefly, cortices are rapidly removed following decapitation of carbon dioxide-anesthetized Sprague-Dawley rats (200-250 g). The cortices are homogen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2PZ5D0BUS Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482692(CHEMBL390326)copy SMILEScopy InChI
Affinity DataIC50: 20nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM238234(US9388210, 14a | US9388210, 6a)copy SMILEScopy InChI
Affinity DataIC50: 25nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4949US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM238243(US9388210, 16a)copy SMILEScopy InChI
Affinity DataIC50: 28nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4949US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540749(US11261211, Compound SA-12)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540750(US11261211, Compound SA-20)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540751(US11261211, Compound SA-22)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540752(US11261211, Compound SA-13)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540755(US11261211, Compound SA-10 | US11261211, Compound ...)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540756(US11261211, Compound SA-54)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540758(US11261211, Compound SA-40)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540747(US11261211, Compound SA-23)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540746(US11261211, Compound SA-21)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540745(US11261211, Compound SA-19)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540744(US11261211, Compound SA-18)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540743(US11261211, Compound SA-17)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540742(US11261211, Compound SA-16)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540741(US11261211, Compound SA-5)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540740(US11261211, Compound SA-6)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540739(US11261211, Compound SA-8)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540738(US11261211, Compound SA-7)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540737(US11261211, Compound SA-3)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540734(US11261211, Compound SA-1)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM655561(US11912737, Example 1 | US11912737, Example 7.)copy SMILES
Affinity DataIC50: 30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482694(CHEMBL229535)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482688(CHEMBL387958)copy SMILEScopy InChI
Affinity DataIC50: 30nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540773(US11261211, Compound SB-15)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM655581(US11912737, Example 31.)copy SMILES
Affinity DataIC50: 30nMMore data for this Ligand-Target Pair
Ligand Info
In DepthDetails
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540776(US11261211, Compound SB-45)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540765(US11261211, Compound SA-56)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540799(Compound SA-51 | US11261211, Compound SA-53)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540760(US11261211, Compound SB-49)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540761(US11261211, Compound SB-50)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1(Rattus norvegicus (Rat))TBA
LigandPNGBDBM540755(US11261211, Compound SA-10 | US11261211, Compound ...)copy SMILES
Affinity DataIC50: 30nMAssay Description:TBPS binding assays using rat brain cortical membranes in the presence of 5 μM GABA has been described (Gee et al, J. Pharmacol. Exp. Ther. 1987...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q2988B61US Patent
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50215531(2-chloro-alpha-[[(4-chlorophenyl)amino]methylene]-...)copy SMILEScopy InChI
Affinity DataIC50: 40nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482691(CHEMBL556727)copy SMILEScopy InChI
Affinity DataIC50: 45nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50482690(CHEMBL229374)copy SMILEScopy InChI
Affinity DataIC50: 50nMAssay Description:Inhibition of rat GABA alpha-1-beta-2-gamma-2 receptorMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q27D2XZDPubMed
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-2/gamma-2(Rattus norvegicus (Rat))
Wuhan Institute of Technology

Curated by ChEMBL
LigandPNGBDBM238245(US9388210, 17a)copy SMILEScopy InChI
Affinity DataIC50: 53nMpH: 7.4 T: 2°CAssay Description:Briefly, aliquots of membrane solution (0.5 mg/mL final protein concentration in assay) were incubated with 5 μM GABA, 2 nM [35S]TBPS (45−...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails
BindingDB Entry DOI: 10.7270/Q29K4949US Patent
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