Compile Data Set for Download or QSAR
Found 4 of ic50 for UniProtKB: P63142
TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 5.40E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)3/Kv1.2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 5.70E+4nMAssay Description:Inhibition of recombinant rat Kv(1.1)2/Kv(1.2)2 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed
TargetPotassium voltage-gated channel subfamily A member 2(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.2(4) expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed
TargetPotassium voltage-gated channel subfamily A member 1/2(Rattus norvegicus)
Dublin Institute of Technology

Curated by ChEMBL
LigandPNGBDBM50237157(CHEMBL4079366)copy SMILEScopy InChI
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant rat Kv1.1/Kv(1.2)3 expressed in HEK293 cells at -90 mV holding potential by whole cell patch clamp Qpatch methodMore data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q29K4DHGPubMed