Affinity DataEC50: 0.100nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
Affinity DataEC50: 0.200nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
Affinity DataEC50: 0.220nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig illeum assessed as electric field-stimulated responseMore data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Binding affinity towards k-opioid receptor k-EL-2 mutant (wild-type) expressed in HEK cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 21nMAssay Description:Agonist activity at KOR in guinea pig vas deferensMore data for this Ligand-Target Pair
Affinity DataEC50: 53nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig brain membranes by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 230nMAssay Description:Agonist activity at kappa opioid receptor in guinea pig brain membranes by [35S]-GTPgammaS binding assayMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+3nMAssay Description:Agonist activity at kappa opioid receptor guinea pig colon tissueMore data for this Ligand-Target Pair